Compile Data Set for Download or QSAR
maximum 50k data
Found 27 of ic50 for monomerid = 50181441
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of oseltamivir-resistant Influenza A virus A/WSN/1933(H1N1) recombinant wild type neuraminidase transfected in HEK293 cells using MUNANA a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase expressed in HEK293 cells pre-incubated for 10 mins before 4-M...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of oseltamivir-resistant Influenza A virus A/Vietnam/1194/2004(H5N1) recombinant wild type neuraminidase transfected in HEK293 cells using...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of Influenza A virus (A/WSN/1933(H1N1)) recombinant neuraminidase expressed in HEK293 cells pre-incubated for 10 mins before 4-MUNANA subs...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (strain A/Wilson-Smith/1933 H1N1...)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  0.480nMAssay Description:Inhibition of Influenza A virus (A/WSN/1933(H1N1)) neuraminidase pre-incubated for 10 mins before 4-MUNANA substrate addition by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of Influenza A virus A/Brisbane/10/2007(H3N2) recombinant wild type neuraminidase transfected in HEK293 cells using MUNANA as substrate as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of Influenza A virus A/Shanghai/01/2014(H7N9) recombinant wild type neuraminidase transfected in HEK293 cells using MUNANA as substrate as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (strain A/Memphis/1/1971 H3N2))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  2nMAssay Description:Inhibition of Influenza A virus (A/Brisbane/10/2007(H3N2)) recombinant neuraminidase expressed in HEK293 cells pre-incubated for 10 mins before 4-MUN...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of oseltamivir-resistant Influenza A virus A/Vietnam/1194/2004(H5N1) recombinant neuraminidase H275Y mutant transfected in HEK293 cells us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of Influenza A virus (A/WSN/1933(H1N1)) recombinant neuraminidase H275Y mutant expressed in HEK293 cells pre-incubated for 10 mins before ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of Influenza A virus A/WSN/1933(H1N1) recombinant neuraminidase H275Y mutant transfected in HEK293 cells using MUNANA as substrate assesse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  18nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase H275Y mutant expressed in HEK293 cells pre-incubated for 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  23nMAssay Description:Inhibition of Influenza A virus (A/WSN/1933(H1N1)) neuraminidase H275Y mutant pre-incubated for 10 mins before 4-MUNANA substrate addition by fluorom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  93nMAssay Description:Inhibition of Influenza A virus (A/Shanghai/01/2014(H7N9)) recombinant neuraminidase R292K mutant expressed in HEK293 cells pre-incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  146nMAssay Description:Inhibition of Influenza A virus A/Brisbane/10/2007(H3N2) recombinant neuraminidase R292K mutant transfected in HEK293 cells using MUNANA as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  146nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase R292K mutant expressed in HEK293 cells pre-incubated for 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  225nMAssay Description:Inhibition of Influenza A virus A/Brisbane/10/2007(H3N2) recombinant neuraminidase E119A mutant transfected in HEK293 cells using MUNANA as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  451nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase E119A mutant expressed in HEK293 cells pre-incubated for 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of influenza virus neuraminidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase(Clostridium perfringens)
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  3.96E+4nMAssay Description:Inhibition of Clostridium perfringenes neuraminidase activity using 4-methylumbelliferyl-1-alpha-D-N-acetylneuramic acid sodium salt hydrate as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-2(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of MBP-fused recombinant human neuraminidase 2 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed...More data for this Ligand-Target Pair
TargetSialidase-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human NEU3More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSialidase-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human NEU1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSialidase-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of MBP-fused recombinant human neuraminidase 3 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of recombinant His6-tagged human neuraminidase 1 expressed in HEK293 cells using 4MU-NANA as substrate preincubated for 15 mins followed b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human NEU4More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSialidase-4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of MBP-fused recombinant human neuraminidase 4 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed