Affinity DataIC50: 24nMAssay Description:Antagonist activity at human CysLT1 receptor expressed in Syrian hamster AV12-664 cells assessed as decrease in LTD4-induced intracellular calcium le...More data for this Ligand-Target Pair
Affinity DataIC50: >8.00E+3nMAssay Description:Antagonist activity at recombinant human mGlu1 receptor expressed in hamster AV12 cells expressing EAAT1 assessed as inhibition of glutamate-induced ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.25E+4nMAssay Description:Antagonist activity at recombinant human mGlu5 receptor expressed in hamster AV12 cells expressing EAAT1 assessed as inhibition of glutamate-induced ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.25E+4nMAssay Description:Antagonist activity at recombinant human mGlu2 receptor expressed in hamster AV12 cells expressing EAAT1 assessed as inhibition of glutamate-induced ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.25E+4nMAssay Description:Antagonist activity at recombinant human mGlu3 receptor expressed in hamster AV12 cells expressing EAAT1 assessed as inhibition of glutamate-induced ...More data for this Ligand-Target Pair