Affinity DataIC50: 1.80E+3nMAssay Description:Binding affinity to DP2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetMAP kinase-activated protein kinase 5(Homo sapiens (Human))
Metabasis Therapeutics
Curated by ChEMBL
Metabasis Therapeutics
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PRAK expressed in baculovirus infected Sf21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Reversible inhibition of CYP2D6 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Reversible inhibition of CYP3A4 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >8.60E+4nMAssay Description:Binding affinity to DP2 receptor (unknown origin) in presence of 10% human serumMore data for this Ligand-Target Pair