Affinity DataEC50: 49nMAssay Description:Displacement of [3H]R1881 from AR in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 915nMAssay Description:Displacement of [3H]R1881 from AR in human LNCaP cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 420nMAssay Description:Antagonist activity at full length human androgen receptor expressed in mammalian expression system measured after 22 to 24 hrs by luciferase reporte...More data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Inhibition of DHT-induced androgen receptor transactivation in human LNCaP cells after 24 hrs by luciferase reporter gene assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP C4-2 cells transfected with PSA6.1-luc and pRL-TK measured by luciferase gene reporter assayMore data for this Ligand-Target Pair
Affinity DataEC50: 62nMAssay Description:Agonist activity at VP16-AR F877L mutant (unknown origin) transfected in human HepG2 cells cotransfected with ARE-LUC incubated for 48 hrs by steady-...More data for this Ligand-Target Pair
Affinity DataEC50: 1.14E+4nMAssay Description:Agonist activity at full length androgen receptor F877L mutant (unknown origin) expressed in PC-3 cells assessed as transcriptional activityMore data for this Ligand-Target Pair
Affinity DataEC50: 1.07E+3nMAssay Description:Agonist activity at full length androgen receptor F876L/T877A mutant (unknown origin) expressed in PC-3 cells assessed as transcriptional activityMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Antagonist activity at androgen receptor in human C4-2-PSA-rl cells incubated for 24 hrs in presence of androgen R1881 by dual-glo luciferase reporte...More data for this Ligand-Target Pair