Affinity DataKi: 5.5nMAssay Description:Inhibition of human recombinant DPP4 using Gly-Pro-7-amido-4-methylcoumarin hydrobromide as substrate incubated for 30 mins by fluorescence microplat...More data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Inhibition of human GCGR receptorMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Competitive inhibition of PTP1B (unknown origin) assessed as inhibition constant using pNPP as substrate by Michaelis-Menten based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+4nMAssay Description:Inhibition of human recombinant DPP9 using Gly-Pro-7-amido-4-methylcoumarin hydrobromide as substrate incubated for 30 mins by fluorescence microplat...More data for this Ligand-Target Pair
Affinity DataKi: 3.75E+4nMAssay Description:Inhibition of human recombinant DPP8 using Gly-Pro-7-amido-4-methylcoumarin hydrobromide as substrate incubated for 30 mins by fluorescence microplat...More data for this Ligand-Target Pair