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Found 21 of ic50 for UniProtKB: P28471
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235902(US9365502, MQ-87)
Affinity DataIC50:  14nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235905(US9365502, MQ-85)
Affinity DataIC50:  29nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235901(US9365502, MQ-86)
Affinity DataIC50:  43nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235900(US9365502, MQ-37)
Affinity DataIC50:  46nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235898(US9365502, MQ-38)
Affinity DataIC50:  52nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235894(US9365502, MQ-31)
Affinity DataIC50:  61nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235897(US9365502, MQ-33)
Affinity DataIC50:  62nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235907(US9365502, MQ-39)
Affinity DataIC50:  65nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235896(US9365502, MQ-32)
Affinity DataIC50:  147nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235904(US9365502, MQ-48)
Affinity DataIC50:  282nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4/beta-3/delta(Rattus norvegicus (Rat))
Johannes Gutenberg University Mainz

Curated by ChEMBL
LigandPNGBDBM50457439(CHEMBL4213357)
Affinity DataIC50:  510nMAssay Description:Displacement of [3H]EBOB from rat GABA-A receptor alpha4beta3delta expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235899(US9365502, MQ-83)
Affinity DataIC50:  748nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235910(US9365502, MQ-50)
Affinity DataIC50:  1.06E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235903(US9365502, MQ-47)
Affinity DataIC50:  1.33E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235906(US9365502, MQ-49)
Affinity DataIC50:  1.58E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235895(US9365502, MQ-36)
Affinity DataIC50:  1.73E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4/beta-3(Rattus norvegicus (Rat))
Johannes Gutenberg University Mainz

Curated by ChEMBL
LigandPNGBDBM50457439(CHEMBL4213357)
Affinity DataIC50:  1.86E+3nMAssay Description:Displacement of [3H]EBOB from rat GABA-A receptor alpha4beta3 expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235911(US9365502, MQ-54)
Affinity DataIC50:  1.99E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4/beta-3/gamma-2(Rattus norvegicus (Rat))
Johannes Gutenberg University Mainz

Curated by ChEMBL
LigandPNGBDBM50457439(CHEMBL4213357)
Affinity DataIC50:  3.29E+3nMAssay Description:Displacement of [3H]EBOB from rat GABA-A receptor alpha4beta3gamma2 expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235908(US9365502, MQ-53)
Affinity DataIC50:  3.63E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
Washington University

US Patent
LigandPNGBDBM235909(US9365502, MQ-51)
Affinity DataIC50:  5.86E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent