Affinity DataKd: 0.420nMAssay Description:Binding affinity for membrane-bound 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor in rat cortex using [3H]- ketanserinMore data for this Ligand-Target Pair
Affinity DataKd: >5.01E+3nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor in rat cortex using [3H]- ketanserinMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 0.110nMAssay Description:Binding affinity to rat frontal cortex 5-HT2A assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 1.04nMAssay Description:Compound was tested for its effect on 5-hydroxytryptamine 2 receptor saturation analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptor in membranes of N1E-115 neuroblastoma cells using [3H]-ICS 205-930; Not determinedMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 631nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptor in membranes of N1E-115 neuroblastoma cells using [3H]-ICS 205-930More data for this Ligand-Target Pair
Affinity DataKd: 0.963nMAssay Description:Compound was tested for its effect on 5-hydroxytryptamine 2 receptor saturation analysisMore data for this Ligand-Target Pair