Compile Data Set for Download or QSAR
maximum 50k data
Found 98 of ki for UniProtKB: P35353
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087556((4-Fluoro-butyl)-propyl-[2,5,6-trimethyl-7-(2,4,6-...)
Affinity DataKi:  0.910nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074501(Butyl-ethyl-[2,5,6-trimethyl-7-(2,4,6-trimethyl-ph...)
Affinity DataKi:  1nMAssay Description:Affinity for the Corticotropin releasing factor receptor 1 (CRHR1) was determined in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074439(1-(2-Bromo-4,6-dimethoxy-phenyl)-4,6-dimethyl-1H-p...)
Affinity DataKi:  1nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50058163(Butyl-[2,5-dimethyl-7-(2,4,6-trimethyl-phenyl)-7H-...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50131716(CHEMBL430892 | [3-(4-Bromo-2-chloro-phenyl)-2,5-di...)
Affinity DataKi:  1.90nMAssay Description:Affinity for the Corticotropin releasing factor receptor 1 (CRHR1) was determined in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087559(CHEMBL164206 | Cyclopropylmethyl-propyl-[2,5,6-tri...)
Affinity DataKi:  2.30nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074501(Butyl-ethyl-[2,5,6-trimethyl-7-(2,4,6-trimethyl-ph...)
Affinity DataKi:  2.5nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50096721(5-Chloro-N-cyclopropylmethyl-N'-(2,6-dichloro-4-tr...)
Affinity DataKi:  3nMAssay Description:Binding affinity towards Corticotropin releasing hormone receptor type 1 of rat cerebellum using [125I]-Tyr-sauvagine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087560(CHEMBL348967 | Ethyl-(4-fluoro-butyl)-[2,5,6-trime...)
Affinity DataKi:  3.5nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50116105(3-(6-(dimethylamino)-4-methylpyridin-3-yl)-2,5-dim...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [125I]-sauvagine from rat CRF-1 receptor expressed in rat cortical membrane after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074411((2-Bromo-4,6-dimethoxy-phenyl)-(4,6-dimethyl-pyrim...)
Affinity DataKi:  5nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50348782(CHEMBL1807053)
Affinity DataKi:  9.80nMAssay Description:Displacement of [125I]-sauvagine from rat CRF-1 receptor expressed in rat cortical membrane after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087561(Butyl-(4-fluoro-butyl)-[2,5,6-trimethyl-7-(2,4,6-t...)
Affinity DataKi:  10nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50096722(5-Chloro-N-cyclopropylmethyl-N'-(2,6-dichloro-4-io...)
Affinity DataKi:  14nMAssay Description:Binding affinity towards Corticotropin releasing hormone receptor type 1 of rat cerebellum using [125I]-Tyr-sauvagine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074456(CHEMBL10504 | SC241 | [3-(2-Bromo-4-isopropyl-phen...)
Affinity DataKi:  14.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM85397(CRA1000)
Affinity DataKi:  15.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50177574(3-(4-(2-methoxybenzyloxy)phenylsulfonyl)-N-mesityl...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM85398(CRA1001)
Affinity DataKi:  18.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM85397(CRA1000)
Affinity DataKi:  20.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074456(CHEMBL10504 | SC241 | [3-(2-Bromo-4-isopropyl-phen...)
Affinity DataKi:  20.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50096723(CHEMBL113333 | N-(4-Bromo-2,6-dichloro-phenyl)-5-c...)
Affinity DataKi:  21nMAssay Description:Binding affinity towards Corticotropin releasing hormone receptor type 1 of rat cerebellum using [125I]-Tyr-sauvagine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074372((2-Bromo-4-isopropyl-phenyl)-ethyl-(4-methyl-6-mor...)
Affinity DataKi:  22nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM85398(CRA1001)
Affinity DataKi:  22.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074435(1-(2-Bromo-4-isopropyl-phenyl)-6-methyl-4-morpholi...)
Affinity DataKi:  28nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074420(1-(2-Bromo-4,6-dimethoxy-phenyl)-4,6-dimethyl-1H-p...)
Affinity DataKi:  29nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087557(CHEMBL164042 | Cyclopropylmethyl-(3-fluoro-propyl)...)
Affinity DataKi:  30nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50054245(5-Chloro-N-cyclopropylmethyl-2-methyl-N-propyl-N''...)
Affinity DataKi:  31nMAssay Description:Binding affinity towards Corticotropin releasing hormone receptor type 1 of rat cerebellum using [125I]-Tyr-sauvagine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50177568(3-(4-(benzyloxy)phenylsulfonyl)-N-mesityl-6-methyl...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50177576(3-(4-(3,5-dimethoxybenzyloxy)phenylsulfonyl)-N-mes...)
Affinity DataKi:  34nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074425(1-(2-Bromo-4-isopropyl-phenyl)-6-methyl-4-phenyl-1...)
Affinity DataKi:  34nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074429(1-(2-Bromo-4-isopropyl-phenyl)-6-methyl-4-phenyl-1...)
Affinity DataKi:  36nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074351((4,6-Dimethyl-pyrimidin-2-yl)-ethyl-(2-iodo-4-isop...)
Affinity DataKi:  38nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074351((4,6-Dimethyl-pyrimidin-2-yl)-ethyl-(2-iodo-4-isop...)
Affinity DataKi:  38nMAssay Description:Binding affinity of the compound was measured on rat Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074353((2-Bromo-4,6-dimethoxy-phenyl)-ethyl-(4-methyl-6-m...)
Affinity DataKi:  43nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074350((2-Bromo-4-isopropyl-phenyl)-(4,6-dimethyl-pyrimid...)
Affinity DataKi:  46nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074350((2-Bromo-4-isopropyl-phenyl)-(4,6-dimethyl-pyrimid...)
Affinity DataKi:  46nMAssay Description:Binding affinity of the compound was measured on rat Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074437(1-(2-Bromo-4-isopropyl-phenyl)-4,6-dimethyl-1H-pyr...)
Affinity DataKi:  47nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074432((4,6-Dimethyl-pyrimidin-2-yl)-(2-iodo-4-isopropyl-...)
Affinity DataKi:  48nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50177581(CHEMBL437893 | methyl 3-((4-(2-(mesitylamino)-6-me...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50177584(3-(4-ethylphenylsulfonyl)-N-mesityl-6-methylpyridi...)
Affinity DataKi:  52nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50177572(3-(4-(3-methoxybenzyloxy)phenylsulfonyl)-N-mesityl...)
Affinity DataKi:  58nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074430(1-(2-Bromo-4-isopropyl-phenyl)-4-chloro-6-methyl-1...)
Affinity DataKi:  67nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50177582(3-((4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfon...)
Affinity DataKi:  75nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074419(1-(2-Bromo-4-isopropyl-phenyl)-6-chloro-4-methyl-1...)
Affinity DataKi:  79nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074408((2-Bromo-4-isopropyl-phenyl)-(4,6-dimethyl-pyrimid...)
Affinity DataKi:  96nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074408((2-Bromo-4-isopropyl-phenyl)-(4,6-dimethyl-pyrimid...)
Affinity DataKi:  96nMAssay Description:Binding affinity of the compound was measured on rat Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50403726(CHEMBL2112936)
Affinity DataKi:  110nMAssay Description:Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074423(1-(2-Bromo-4-isopropyl-phenyl)-6-methyl-4-morpholi...)
Affinity DataKi:  112nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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