Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ki for UniProtKB: P56817
TargetBeta-secretase 1 [22-457](Homo sapiens (Human))
Philipps University Marburg

LigandPNGBDBM32389(phenyl-substituted sulfonamides, 6f)
Affinity DataKi:  6.40E+4nM ΔG°:  -5.72kcal/moleT: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1 [22-457](Homo sapiens (Human))
Philipps University Marburg

LigandPNGBDBM32386(phenyl-substituted sulfonamides, 6c)
Affinity DataKi:  1.50E+5nM ΔG°:  -5.21kcal/moleT: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed