Affinity DataEC50: 0.191nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.257nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 0.324nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 0.324nMAssay Description:Agonist activity at A2BR in human NHVCF cells assessed as cAMP accumulation incubated for 30 mins by LANCE cAMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.380nMAssay Description:Agonist activity at human A2B receptor expressed in Flp-In-CHO cells assessed as cAMP accumulation incubated for 10 mins in presence of forskolin by ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.389nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.468nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 0.501nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.692nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 0.871nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 2.20nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as increase in intracellular cAMP level after 30 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 3.40nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.5nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.80nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.90nMpH: 7.4 T: 2°CAssay Description:The following test protocol is used for pharmacologically characterizing
cells and for the robot-assisted substance screening:The stock cultures
ar...More data for this Ligand-Target Pair
Affinity DataEC50: 4.60nMAssay Description:Agonist activity at human A2B receptor expressed in Flp-In-CHO cells assessed as cAMP accumulation incubated for 10 mins in presence of forskolin by ...More data for this Ligand-Target Pair
Affinity DataEC50: 4.80nMAssay Description:Agonist activity at human A2B receptor expressed in Flp-In-CHO cells assessed as cAMP accumulation incubated for 10 mins in presence of forskolin by ...More data for this Ligand-Target Pair
Affinity DataEC50: 4.90nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.5nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.80nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Agonist activity at human A2B receptor expressed in Flp-In-CHO cells assessed as cAMP accumulation incubated for 10 mins in presence of forskolin by ...More data for this Ligand-Target Pair
Affinity DataEC50: 7.30nMAssay Description:Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 7.40nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 7.40nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Agonistic activity against human adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 9.5nMAssay Description:Agonist activity at human adenosine A2B receptor expressed in CHO cell membranes assessed as induction of cAMP accumulation by AlphaScreen assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.5nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 9.80nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: <10nMAssay Description:Stably transfected HEK-293 cells expressing the human adenosine A2B receptor (Perkin Elmer) were maintained in MEM culture medium with 10% FBS and 10...More data for this Ligand-Target Pair
Affinity DataEC50: <10nMAssay Description:Stably transfected HEK-293 cells expressing the human adenosine A2B receptor (Perkin Elmer) were maintained in MEM culture medium with 10% FBS and 10...More data for this Ligand-Target Pair
Affinity DataEC50: <10nMAssay Description:Stably transfected HEK-293 cells expressing the human adenosine A2B receptor (Perkin Elmer) were maintained in MEM culture medium with 10% FBS and 10...More data for this Ligand-Target Pair
Affinity DataEC50: <10nMAssay Description:Stably transfected HEK-293 cells expressing the human adenosine A2B receptor (Perkin Elmer) were maintained in MEM culture medium with 10% FBS and 10...More data for this Ligand-Target Pair
Affinity DataEC50: <10nMAssay Description:Stably transfected HEK-293 cells expressing the human adenosine A2B receptor (Perkin Elmer) were maintained in MEM culture medium with 10% FBS and 10...More data for this Ligand-Target Pair