Affinity DataKi: 1.30nMAssay Description:Binding affinity to rat 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity to rat 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 186nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 239nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 379nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 388nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 431nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 506nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 736nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 752nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 998nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]-LSD as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]-LSD as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]-LSD as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]-LSD as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.50E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]-LSD as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]-LSD as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >6.40E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]-LSD as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7(Rattus norvegicus)
Solvay Duphar
Curated by ChEMBL
Solvay Duphar
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity was measured on 5-hydroxytryptamine receptor uptake receptor using [3H]- paroxetine as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7(Rattus norvegicus)
Solvay Duphar
Curated by ChEMBL
Solvay Duphar
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]- GR-65,630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of specific [3H]-OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair