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maximum 50k data
Found 89 of ic50 for UniProtKB: P21729
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040317(CHEMBL262756 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50:  0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040299(CHEMBL410783 | cyclopropylbenzene(CO)His-Trp-Ala-V...)
Affinity DataIC50:  0.0300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040325(CHEMBL268386 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  0.0380nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040299(CHEMBL410783 | cyclopropylbenzene(CO)His-Trp-Ala-V...)
Affinity DataIC50:  0.0490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50:  0.0500nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50:  0.0500nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)
Affinity DataIC50:  0.0790nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040308(2-aminoPhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50:  0.100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50:  0.160nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040315((CH3)2PhC(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe...)
Affinity DataIC50:  0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040315((CH3)2PhC(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe...)
Affinity DataIC50:  0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040317(CHEMBL262756 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  0.220nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50:  0.230nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)
Affinity DataIC50:  0.300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040320(CHEMBL264122 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  0.330nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407275(CHEMBL2112786)
Affinity DataIC50:  0.490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040316(3-isoquinolyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50:  0.570nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012304(2-{2-[2-[2-(2,2-Dimethyl-propionylamino)-3-(3H-imi...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040324(CHEMBL266516 | PhCH2CH2(CO)His-(BzthAla)-Ala-Val-D...)
Affinity DataIC50:  0.75nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)
Affinity DataIC50:  1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)
Affinity DataIC50:  1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407273(CHEMBL2111953)
Affinity DataIC50:  1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50:  1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040314((CH3)2PhCCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50:  1.20nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012313(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50:  1.20nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407273(CHEMBL2111953)
Affinity DataIC50:  1.30nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012318(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012304(2-{2-[2-[2-(2,2-Dimethyl-propionylamino)-3-(3H-imi...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012306(Ac-His-Trp-Ala-Val-Gly-His-Leu-Met-NH2 | CHEMBL274...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040323(CHEMBL265736 | phenothiazoneCH2CH2(CO)His-Trp-Ala-...)
Affinity DataIC50:  1.90nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012317(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50:  2nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040298(CHEMBL386478 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  2nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040308(2-aminoPhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50:  2nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012311(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012307(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012308(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012318(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50:  3nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407277(CHEMBL2112785)
Affinity DataIC50:  3nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407277(CHEMBL2112785)
Affinity DataIC50:  3nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012309(Ac-His-Trp-Ala-Val-D-Ala-His-Leu-Met-NH2 | CHEMBL2...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012297(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50:  3.30nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040319(4-CF3PhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50:  3.70nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012300(2-[2-[2-(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012317(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50:  4nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012314((CH3)CCO-His-Trp-Ala-Val-Gly-His-Leu-Met-NH2 | CHE...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012312(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012319(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50:  5nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040298(CHEMBL386478 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)
Affinity DataIC50:  5nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040304(CHEMBL267943 | PhCH2CH2(CO)ThiAla-Trp-Ala-Val-DAla...)
Affinity DataIC50:  5.60nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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