Compile Data Set for Download or QSAR
maximum 50k data
Found 51 of ki for UniProtKB: P52500
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50408923(CHEMBL2114155)
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50005601(CHEMBL2369819)
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85480((3-Ph-Pr6)His7,DAla11,DPro13,Psi13-14,Phe14-Bn(6-1...)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85500(Bombesin,Phe13)
Affinity DataKi:  0.770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  0.990nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089280(CHEMBL437655 | JMV 1535)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089284(CHEMBL265856 | JMV 1803)
Affinity DataKi:  1.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85499(CAS_29451-71-6 | NSC_5489061 | Ranatensin)
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85486(DPhe6-Bn[6-14))
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85502(PG-L)
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089285(CHEMBL415110 | JMV 1799)
Affinity DataKi:  3.10nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089282((D)Phe-Gln-Trp-Ala-Val-Gly-His-Leu-Leu-NH2 | CHEMB...)
Affinity DataKi:  3.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089281(CHEMBL386480 | JMV 1802)
Affinity DataKi:  3.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089291(CHEMBL415021 | JMV 1813)
Affinity DataKi:  5.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85498(CAS_5486808 | Litorin | NSC_5486808)
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85495(DPhe6-Bn(6-13)propylamide)
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85493(DTyr6,DAla11-Bn(6-13)butylamide)
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089278(CHEMBL411016 | JMV 1801)
Affinity DataKi:  9nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85496(DPhe6-Bn(6-13)methylester)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089279(CHEMBL406013 | JMV 1719)
Affinity DataKi:  13nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85481(CAS_93755-85-2 | GRP)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM81964(CAS_5486814 | Gastrin | NSC_5486814 | Neuromedin C)
Affinity DataKi:  20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85494(DPhe6-Bn(6-13)NH2)
Affinity DataKi:  27nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85506(CAS_125988 | NSC_125988 | Rhodei-Litorin)
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85490(DPhe6,Leu13,Psi(CH2NH),Cpa14-Bn(6-14))
Affinity DataKi:  42nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85497(Alytesin | CAS_31078-12-3)
Affinity DataKi:  62nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85482(DPhe6-Bn(6-13)hexylamide)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089286(CHEMBL407022 | JMV 1693)
Affinity DataKi:  127nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85492(GRP-10,frog)
Affinity DataKi:  130nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  180nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50408922(CHEMBL2115179)
Affinity DataKi:  225nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85483(CAS_5748287 | NSC_5748287 | Phyllolitorin)
Affinity DataKi:  240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  248nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089288(Bombesin analogues | CHEMBL415022)
Affinity DataKi:  300nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85487(Leu8-phyllolitorin)
Affinity DataKi:  420nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85491(Leu13,Psi(CH2NH),Leu14-BN)
Affinity DataKi:  430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85489(DPhe6,12,Leu14-Bn)
Affinity DataKi:  430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85479(DPhe6-Bn(1-13)NH2)
Affinity DataKi:  450nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089292(Bombesin analogues | CHEMBL439440)
Affinity DataKi:  500nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089290(Bombesin analogues | CHEMBL413938)
Affinity DataKi:  650nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85501(DPhe6-Bn(6-13)hydrazide)
Affinity DataKi:  1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089293(Bombesin analogues | CHEMBL407481)
Affinity DataKi:  2.25E+3nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85485(DPhe6-Bn(6-13)NHN(ME)2)
Affinity DataKi:  3.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85478(Bombesin, SAP | CAS_31362-50-2)
Affinity DataKi:  3.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85504(Substance P,[DArg1,DTrp7,9,Leu11])
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85503(Dphe12-Bn)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50063814(CHEMBL217438 | Dnal,Cys,Tyr,DTrp,Lys,Val,Cys,Nal-n...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85505(Substance P(4-11),[Dpro4,Dtrp7,9,10])
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089287(Bombesin analogues | CHEMBL384242)
Affinity DataKi: >1.00E+6nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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