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Found 10 of ki for UniProtKB: P16233
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))TBA
LigandPNGBDBM50212744(CHEBI:35020 | TRIBUTYRIN)
Affinity DataKi: <1nM Kon:  1M-1s-1Assay Description:Tested for hydrolysis with 0.2 ug/mL of PPL (porcine pancreatic lipase), 1.5 ug/mL of colipase and 4 mM sodium taurodeoxycholatet (NaTDC) at a compou...More data for this Ligand-Target Pair
In DepthDetails
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))TBA
LigandPNGBDBM50212746(CHEMBL119630)
Affinity DataKi:  220nM Kon:  220M-1s-1Assay Description:Tested for hydrolysis with 0.5 ug/mL of PPL (porcine pancreatic lipase), 1.5 ug/mL of colipase and 4 mM of sodium taurodeoxycholatet (NaTDC) at the c...More data for this Ligand-Target Pair
In DepthDetails
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))TBA
LigandPNGBDBM50212746(CHEMBL119630)
Affinity DataKi:  710nM Kon:  710M-1s-1Assay Description:Tested for hydrolysis with 1.0 ug/mL of PPL (porcine pancreatic lipase), 2.2 ug/mL of colipase and 4 mM of sodium taurodeoxycholatet (NaTDC) at the c...More data for this Ligand-Target Pair
In DepthDetails
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))TBA
LigandPNGBDBM50212744(CHEBI:35020 | TRIBUTYRIN)
Affinity DataKi:  1.10E+3nM Kon:  1.10E+3M-1s-1Assay Description:Tested for hydrolysis with 0.2 ug/mL of PPL (porcine pancreatic lipase) at a compound dose of 0.2 gMore data for this Ligand-Target Pair
In DepthDetails
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))TBA
LigandPNGBDBM50212746(CHEMBL119630)
Affinity DataKi:  2.10E+3nM Kon:  2.10E+3M-1s-1Assay Description:Tested for hydrolysis with 0.2 ug/mL of PPL (porcine pancreatic lipase) at the compound dose of 0.2 gMore data for this Ligand-Target Pair
In DepthDetails
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))TBA
LigandPNGBDBM50212746(CHEMBL119630)
Affinity DataKi:  5.70E+3nM Kon:  5.70E+3M-1s-1Assay Description:Tested for hydrolysis with 1.0 ug/mL of PPL (porcine pancreatic lipase)at the compound dose of 0.2 gMore data for this Ligand-Target Pair
In DepthDetails
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))TBA
LigandPNGBDBM50381861(CHEMBL2022676)
Affinity DataKi:  6.70E+4nMAssay Description:Inhibition of human pancreatic lipase using p-nitrophenylbutyrate as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))TBA
LigandPNGBDBM50381860(CHEMBL2022680)
Affinity DataKi:  1.70E+5nMAssay Description:Inhibition of human pancreatic lipase using p-nitrophenylbutyrate as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))TBA
LigandPNGBDBM50381859(CHEMBL2022681)
Affinity DataKi:  3.60E+5nMAssay Description:Inhibition of human pancreatic lipase using p-nitrophenylbutyrate as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))TBA
LigandPNGBDBM50381858(CHEMBL2022679)
Affinity DataKi:  5.50E+5nMAssay Description:Inhibition of human pancreatic lipase using p-nitrophenylbutyrate as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed