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Found 50 of ic50 for UniProtKB: P33072
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633180(4-((1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-2-methyl...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633249(N-((1-(4-(((1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-...)
Affinity DataIC50: <300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633181(1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-3-(3-(N,N-di...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633197(N,N′-((((((((((5-(1-((Z)-4-amino-2-fluorobut...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633202(N,N′-((((5-(1-((Z)-4-amino-2-fluorobut-2-en-...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633250(N-((1-(4-(((1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633203(5-(1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-3-(3-(N,N...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633204(5-(4-(1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-3-(3-(...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633224(4-(((Z)-4-amino-2-fluorobut-2-en-1-yl)sulfonyl)-N-...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633227(2-(((Z)-4-amino-2-fluorobut-2-en-1-yl)sulfonyl)-N-...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633233(3-(((Z)-4-amino-2-fluorobut-2-en-1-yl)sulfonyl)-N-...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633244(3-(((Z)-4-amino-2-fluorobut-2-en-1-yl)sulfonyl)-N-...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633245((3aS,4S,6aR)-4-(5-(4-(3-(3-(((Z)-4-amino-2-fluorob...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633246((3aS,3a'S,4S,4'S,6aR,6a′R)-4,4′-(((((5...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633247((3aS,3a'S,4S,4'S,6aR,6a′R)-4,4′-(((((3...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM633248((3aS,4S,6aR)-4-(4-(4-(3-((3-(((Z)-4-amino-2-fluoro...)
Affinity DataIC50: >300nMAssay Description:The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the isoenz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505649(CHEMBL4439437)
Affinity DataIC50:  398nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505633(CHEMBL4448713)
Affinity DataIC50:  398nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505657(CHEMBL4467234)
Affinity DataIC50:  501nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505655(CHEMBL4441299)
Affinity DataIC50:  501nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505659(CHEMBL4459524)
Affinity DataIC50:  501nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505650(CHEMBL4450939)
Affinity DataIC50:  631nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505640(CHEMBL4556859)
Affinity DataIC50:  631nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505641(CHEMBL4531248)
Affinity DataIC50:  794nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505661(CHEMBL4574820)
Affinity DataIC50:  794nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505634(CHEMBL4569453)
Affinity DataIC50:  794nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505647(CHEMBL4531065)
Affinity DataIC50:  794nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505660(CHEMBL4581561)
Affinity DataIC50:  794nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505653(CHEMBL4458907)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505636(CHEMBL4443268)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505658(CHEMBL4581458)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505645(CHEMBL4550754)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505643(CHEMBL4582216)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505662(CHEMBL4446643)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  1.78E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  1.78E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505635(CHEMBL4472333)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505648(CHEMBL4562149)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505652(CHEMBL4463296)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505639(CHEMBL4554097)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505637(CHEMBL4438235)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505654(CHEMBL4586209)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505642(CHEMBL4527340)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505651(CHEMBL4469240)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505663(CHEMBL4451632)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505656(CHEMBL4457469)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505646(CHEMBL4446904)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50505644(CHEMBL4563012)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-lysine 6-oxidase(Bos taurus)
Pharmaxis

US Patent
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of bovine aorta LOXMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed