Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ic50 for UniProtKB: P16390
LigandPNGBDBM50115772(CHEMBL3609094)
Affinity DataIC50:  0.0230nMAssay Description:Displacement of [125I]-ChTX from mouse Kv1.3 after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50083523((1-Benzyl-1H-quinolin-4-ylidene)-pentyl-amine | CH...)
Affinity DataIC50:  230nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50098785(4-Benzhydryloxymethyl-1-[3-(4-methoxy-phenyl)-prop...)
Affinity DataIC50:  280nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50098782(2-Isopropyl-8-methoxy-5-methyl-5H-furo[3,2-c]quino...)
Affinity DataIC50:  5.00E+3nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50098781(9-Methoxy-2,2,6-trimethyl-2,6-dihydro-pyrano[3,2-c...)
Affinity DataIC50:  1.00E+4nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50098784(9-Methoxy-2,2,6-trimethyl-2,3,4,6-tetrahydro-pyran...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of voltage-gated potassium channel subunit Kv1.3 expressed in L929 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50098783(4,6,7-Trimethoxy-furo[2,3-b]quinoline | CHEMBL2787...)
Affinity DataIC50:  4.90E+4nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed