Affinity DataEC50: 0.0300nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand Info
Ligand Info
Ligand Info
Ligand Info
3D Structure (crystal)
Ligand Info
Affinity DataEC50: 0.260nMAssay Description:Agonist activity at AhR in human HepG2 cells assessed as induction of CYP1A1 expression after 24 hrs by ethoxyresorufin-O-deethylase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.270nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand Info
Ligand Info
Ligand Info
Affinity DataEC50: 0.340nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand Info
Ligand Info
Affinity DataEC50: 0.440nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.447nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Ligand Info
Ligand Info
Affinity DataEC50: 0.700nMAssay Description:Activation of AhR in human HaCaT cells assessed as induction of XRE-dependent reporter activity incubated for 4 hrs by Renilla/Firefly based dual-luc...More data for this Ligand-Target Pair
Affinity DataEC50: 0.830nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.17nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 1.48nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity at AhR (unknown origin) transfected in human AZ-AHR reporter cells derived from human HepG2 cells incubated for 4 hrs by luciferase ...More data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at AhR in human HepG2 cells assessed as induction of CYP1A1 expression after 24 hrs by ethoxyresorufin-O-deethylase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at AHR in human HepG2 cells incubated for 4.5 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at AHR in human HepG2 cells incubated for 4.5 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Activation of AhR in human HepG2 cells assessed as induction of XRE-dependent reporter activity incubated for 4 hrs by Renilla/Firefly based dual-luc...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Concentration of the compound to bind to human AhR-modied electrodeMore data for this Ligand-Target Pair
Affinity DataEC50: 6.61nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 8.40nMAssay Description:Agonist activity at AhR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 9.60nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 11.5nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Ligand Info
Affinity DataEC50: 15.1nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 15.5nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 17.0nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
Affinity DataEC50: 22.2nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Agonist activity at AhR in human recombinant HepG2-Lucia AhR cell incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 25.1nMAssay Description:Affinity on cytosolic Aromatic hydrocarbon receptor (Ah)More data for this Ligand-Target Pair
