Compile Data Set for Download or QSAR
maximum 50k data
Found 20 of ki for UniProtKB: P22909
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554696(CHEMBL4749860)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50597775(CHEMBL5198566)
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [3H]NECA from A2AAR in rat striata assessed as inhibition constant in presence of N6-cyclopentyladenosine by radioligand competitive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554684(CHEMBL4796664)
Affinity DataKi:  4.70E+3nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554685(CHEMBL4749263)
Affinity DataKi:  5.00E+3nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50597773(CHEMBL4535634)
Affinity DataKi:  5.46E+3nMAssay Description:Displacement of [3H]NECA from A2AAR in rat striata assessed as inhibition constant in presence of N6-cyclopentyladenosine by radioligand competitive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554689(CHEMBL4754656)
Affinity DataKi:  7.10E+3nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50597774(CHEMBL5178192)
Affinity DataKi:  9.92E+3nMAssay Description:Displacement of [3H]NECA from A2AAR in rat striata assessed as inhibition constant in presence of N6-cyclopentyladenosine by radioligand competitive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554691(CHEMBL4764318)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554690(CHEMBL4782649)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554694(CHEMBL4740168)
Affinity DataKi:  1.50E+4nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554692(CHEMBL4751862)
Affinity DataKi:  1.50E+4nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554686(CHEMBL4754362)
Affinity DataKi:  1.50E+4nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50077537((+)-(7-nitro-1,2,3,4-tetrahydroisoquinolin-3-yl)me...)
Affinity DataKi:  1.90E+4nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554695(CHEMBL4760727)
Affinity DataKi:  3.30E+4nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554683(CHEMBL4783068)
Affinity DataKi:  5.20E+4nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554693(CHEMBL4800292)
Affinity DataKi:  6.40E+4nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50597772(CHEMBL5170103)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]NECA from A2AAR in rat striata assessed as inhibition constant in presence of N6-cyclopentyladenosine by radioligand competitive ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554681(CHEMBL4795252)
Affinity DataKi:  1.30E+5nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50023452(1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...)
Affinity DataKi:  2.50E+5nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Rattus norvegicus)
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50294573((2R,3R,4S,5S)-2-(6-amino-9H-purin-9-yl)-5-((2-amin...)
Affinity DataKi:  1.10E+6nMAssay Description:Displacement of [3H]-clonidine from Sprague-Dawley rat alpha2 adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed