Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ic50 for UniProtKB: P19493
TargetGlutamate receptor 4(Rattus norvegicus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50316374(CHEMBL1096289 | N-(4-hydroxyphenylpropanyl)-spermi...)
Affinity DataIC50:  320nMAssay Description:Inhibition of rat recombinant GluA4 receptor expressed in Xenopus oocytes assessed as inhibition of 300 uM kainate-induced currentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50158554(CHEMBL224688 | {2-[3-(3-bromophenyl)ureido]-4-chlo...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50158555(1-[5-chloro-2-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50137125(2-(3-(3-bromophenyl)ureido)-4-chlorobenzoic acid |...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50158561(2-[3-(3-bromophenyl)ureido]-4-chlorobenzenesulfoni...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50137124(4-Chloro-2-(3-naphthalen-2-yl-ureido)-benzoic acid...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Rattus norvegicus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50158556(1-(3-bromophenyl)-3-[5-chloro-2-(1H-tetrazol-5-yl-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed