TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison
Curated by ChEMBL
University Of Wisconsin-Madison
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Compound was evaluated for potency towards nicotinic acetylcholine receptor in rat P2 brain membranes using [3H]-nicotine as a radioligandMore data for this Ligand-Target Pair
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison
Curated by ChEMBL
University Of Wisconsin-Madison
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Inhibition of R. chinensis pepsinMore data for this Ligand-Target Pair
Affinity DataKi: 21nMpH: 7.4Assay Description:The compound was tested for inhibition of rat plasma renin at pH of 7.4.More data for this Ligand-Target Pair
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison
Curated by ChEMBL
University Of Wisconsin-Madison
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Inhibition of R. chinensis pepsinMore data for this Ligand-Target Pair
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison
Curated by ChEMBL
University Of Wisconsin-Madison
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Inhibition of R. chinensis pepsinMore data for this Ligand-Target Pair
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison
Curated by ChEMBL
University Of Wisconsin-Madison
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Inhibition of R. chinensis pepsinMore data for this Ligand-Target Pair
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison
Curated by ChEMBL
University Of Wisconsin-Madison
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Inhibition of R. chinensis pepsinMore data for this Ligand-Target Pair
Affinity DataKi: 115nMpH: 6.0Assay Description:The compound was tested for inhibition of rat plasma renin at pH of 6.0.More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Binding affinity against nicotinic acetylcholine receptor alpha4-beta4 using [3H]epibatidine as radioligand expressed in HEK293 cells or tsA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 230nMpH: 7.4Assay Description:Inhibition of rhizopuspepsinMore data for this Ligand-Target Pair
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison
Curated by ChEMBL
University Of Wisconsin-Madison
Curated by ChEMBL
Affinity DataKi: 336nMAssay Description:Compound was evaluated for inhibitory activity towards nicotinic acetylcholine receptor in rat P2 brain membranes using [3H]-nicotine as a radioligan...More data for this Ligand-Target Pair
Affinity DataKi: 630nMpH: 7.4Assay Description:Binding affinity against nicotinic acetylcholine receptor using [3H]epibatidine as radioligand in rat brain tissueMore data for this Ligand-Target Pair
Affinity DataKi: 630nMpH: 7.4Assay Description:Inhibition of rhizopuspepsinMore data for this Ligand-Target Pair