Compile Data Set for Download or QSAR
maximum 50k data
Found 13 of ki data for polymerid = 50001946,50003274,50006974
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50070005(((3R,6R,15R)-15-Hydroxymethyl-3-isopropyl-2,5-diox...)
Affinity DataKi:  1.30nMAssay Description:Compound was evaluated for potency towards nicotinic acetylcholine receptor in rat P2 brain membranes using [3H]-nicotine as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50022290(2-(3-Hydroxy-6-methyl-4-{3-methyl-2-[3-methyl-2-(3...)
Affinity DataKi:  11nMAssay Description:Inhibition of R. chinensis pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50405190(CHEMBL2028991)
Affinity DataKi:  21nMpH: 7.4Assay Description:The compound was tested for inhibition of rat plasma renin at pH of 7.4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50022287(8-Acetylamino-3-hydroxy-4-{3-methyl-2-[3-methyl-2-...)
Affinity DataKi:  29nMAssay Description:Inhibition of R. chinensis pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50022285((3S,4S) Acetate7-ethoxycarbonyl-6-hydroxy-5-{3-met...)
Affinity DataKi:  33nMAssay Description:Inhibition of R. chinensis pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017789((3S,4S)-3-Hydroxy-6-methyl-4-{3-methyl-2-[3-methyl...)
Affinity DataKi:  42nMAssay Description:Inhibition of R. chinensis pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50022289(Acetate6-ethoxycarbonyl-5-hydroxy-4-{3-methyl-2-[3...)
Affinity DataKi:  47nMAssay Description:Inhibition of R. chinensis pepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50405191(CHEMBL269752)
Affinity DataKi:  115nMpH: 6.0Assay Description:The compound was tested for inhibition of rat plasma renin at pH of 6.0.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rhizopus chinensis)
TBA

Curated by ChEMBL
LigandPNGBDBM50405190(CHEMBL2028991)
Affinity DataKi:  230nMAssay Description:Binding affinity against nicotinic acetylcholine receptor alpha4-beta4 using [3H]epibatidine as radioligand expressed in HEK293 cells or tsA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rhizopus chinensis)
TBA

Curated by ChEMBL
LigandPNGBDBM50405190(CHEMBL2028991)
Affinity DataKi:  230nMpH: 7.4Assay Description:Inhibition of rhizopuspepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRhizopuspepsin(Rhizopus microsporus var. chinensis)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50070006(((Z)-(3R,6R,15R)-15-Hydroxymethyl-3-isopropyl-2,5-...)
Affinity DataKi:  336nMAssay Description:Compound was evaluated for inhibitory activity towards nicotinic acetylcholine receptor in rat P2 brain membranes using [3H]-nicotine as a radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rhizopus chinensis)
TBA

Curated by ChEMBL
LigandPNGBDBM50405191(CHEMBL269752)
Affinity DataKi:  630nMpH: 7.4Assay Description:Binding affinity against nicotinic acetylcholine receptor using [3H]epibatidine as radioligand in rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rhizopus chinensis)
TBA

Curated by ChEMBL
LigandPNGBDBM50405191(CHEMBL269752)
Affinity DataKi:  630nMpH: 7.4Assay Description:Inhibition of rhizopuspepsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed