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Found 31 of ic50 for UniProtKB: P28088
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50043326(CHEMBL438733 | c(Cys-Ser-Cys)-Ser-Ser-Leu-Met-Asp-...)
Affinity DataIC50:  0.0930nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)
Affinity DataIC50:  0.120nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50043322(CHEMBL427748 | c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp...)
Affinity DataIC50:  0.170nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368776(CHEMBL1790962)
Affinity DataIC50:  0.170nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289647(CHEMBL263855 | Compound RES-701-1(1-10)/[A15]ET-1)
Affinity DataIC50:  0.240nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368772(CHEMBL2373291)
Affinity DataIC50:  0.25nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368774(CHEMBL1790963)
Affinity DataIC50:  0.330nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50368777(CHEMBL2373292)
Affinity DataIC50:  0.420nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50043324(CHEMBL411171 | c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp...)
Affinity DataIC50:  0.450nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289650(CHEMBL414047 | Compound RES-701-1(1-10)/[A15]ET-3)
Affinity DataIC50:  2.5nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289648(CHEMBL408437 | Compound RES-701-1(1-10)/[A15]SRTX6...)
Affinity DataIC50:  3.80nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289112(CHEMBL438745 | RES-701-1-C-terminal analogue)
Affinity DataIC50:  6.30nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289108(CHEMBL384792 | RES-701-1 | RES-701-1-C-terminal an...)
Affinity DataIC50:  7.30nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289108(CHEMBL384792 | RES-701-1 | RES-701-1-C-terminal an...)
Affinity DataIC50:  10nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289111(CHEMBL411057 | RES-701-1-C-terminal analogue)
Affinity DataIC50:  10nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289107(CHEMBL263294 | RES-701-1-C-terminal analogue)
Affinity DataIC50:  12nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289113(CHEMBL267754 | RES-701-1-C-terminal analogue)
Affinity DataIC50:  36nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289117(CHEMBL407422 | RES-701-1-C-terminal analogue)
Affinity DataIC50:  45nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289109(CHEMBL409339 | RES-701-1-C-terminal analogue)
Affinity DataIC50:  54nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289116(CHEMBL441573 | RES-701-1-C-terminal analogue)
Affinity DataIC50: >98nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289115(CHEMBL410321 | RES-701-1-C-terminal analogue)
Affinity DataIC50:  120nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289114(CHEMBL409433 | RES-701-1-C-terminal analogue)
Affinity DataIC50:  450nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289110(CHEMBL414131 | RES-701-1-C-terminal analogue)
Affinity DataIC50:  470nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289656(CHEMBL416287 | RES-701-1)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289653(ENDOTHELIN | ET-1 | Endothelin 1 | Et 1)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289651(CHEMBL407188 | Compound [S15]ET-1)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289654(CHEMBL436894 | Compound SRTX6b)
Affinity DataIC50:  3.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289652(CHEMBL437610 | Compound ET-3)
Affinity DataIC50:  3.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289657(CHEMBL414168 | RES-701-1)
Affinity DataIC50:  3.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289655(CHEMBL414740 | N-C cyclized RES-70I-1)
Affinity DataIC50: >5.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Bos taurus)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50289649(CHEMBL429908 | linear peptide of RES-701-1)
Affinity DataIC50:  5.00E+3nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article