Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for UniProtKB: P43219
TargetGastric inhibitory polypeptide receptor(Rattus norvegicus)
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Curated by ChEMBL
LigandPNGBDBM50171817(3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50:  42nMAssay Description:Binding affinity to GIPR in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Rattus norvegicus)
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Curated by ChEMBL
LigandPNGBDBM50202031(3-(4-((1-(4-cyclohexenylphenyl)-3-(3,5-dichlorophe...)
Affinity DataIC50:  216nMAssay Description:Binding affinity to GIPR in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50244455((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3,5-dichl...)
Affinity DataIC50:  501nMAssay Description:Binding affinity to GIPR in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50318666((1R,3S)-5',7-Dichloro-6-fluoro-3-methyl-2,3,4,9-te...)
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity to rat Gip receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed