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Found 14 of ic50 for UniProtKB: P78348
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50096642(CHEMBL3577296)
Affinity DataIC50:  27nMpH: 6.7Assay Description:Inhibition of human ASIC1a endogenously expressed in HEK293 cells clamped at -100 mV gated ionic current at pH 6.7 by standard whole cell patch clamp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50348098(CHEMBL1800430)
Affinity DataIC50:  224nMAssay Description:Inhibition of ASIC1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50408492(CHEMBL5269133)
Affinity DataIC50:  407nMAssay Description:Antagonist activity at human muscarinic acetylcholine M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50408498(CHEMBL5270983)
Affinity DataIC50:  518nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50408502(CHEMBL5289168)
Affinity DataIC50:  729nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50408500(CHEMBL5278611)
Affinity DataIC50:  972nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50408497(CHEMBL5287933)
Affinity DataIC50:  1.42E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50408496(CHEMBL5291421)
Affinity DataIC50:  1.99E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50408493(CHEMBL5285672)
Affinity DataIC50:  1.99E+3nMAssay Description:Antagonist activity at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50408495(CHEMBL5267130)
Affinity DataIC50:  2.59E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50408499(CHEMBL5276647)
Affinity DataIC50:  2.95E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50408494(CHEMBL5267106)
Affinity DataIC50:  3.14E+3nMAssay Description:Antagonist activity at human muscarinic acetylcholine M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50096642(CHEMBL3577296)
Affinity DataIC50:  7.34E+3nMpH: 5.0Assay Description:Inhibition of human ASIC1a endogenously expressed in HEK293 cells clamped at -100 mV gated ionic current at pH 5.0 by standard whole cell patch clamp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute Of Physiology Of Nas Ukraine

Curated by ChEMBL
LigandPNGBDBM50408501(CHEMBL5283083)
Affinity DataIC50:  9.54E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails PubMed