Compile Data Set for Download or QSAR
maximum 50k data
Found 57 of ic50 for UniProtKB: P22612
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  0.700nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50: <1nMAssay Description:Inhibition of PKA (unknown origin) after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human PKAcg using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50587770(CHEMBL5188493)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50228843(CHEMBL436718)
Affinity DataIC50:  3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM3149(2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(4-hydroxybenzen...)
Affinity DataIC50:  4nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  6.5nMAssay Description:In vitro inhibition of Protein Kinase AMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of human PKAcg using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of protein kinase AMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50242733(AT-13148)
Affinity DataIC50: <10nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  15nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM15211(CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...)
Affinity DataIC50:  50nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50587769(CHEMBL5181354)
Affinity DataIC50:  159nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50614310(CHEMBL5269663)
Affinity DataIC50:  184nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50280450(18-hydroxy-3-methoxy-2-methyl-4-methylamino-(2R,3S...)
Affinity DataIC50:  250nMAssay Description:Inhibition of protein kinase AMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50280450(18-hydroxy-3-methoxy-2-methyl-4-methylamino-(2R,3S...)
Affinity DataIC50:  250nMAssay Description:Inhibition of protein kinase AMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50228839(CHEMBL415414)
Affinity DataIC50:  300nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50506921(CHEMBL4459800)
Affinity DataIC50:  790nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50228847(CHEMBL407100)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228846(CHEMBL265876)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM15211(CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of PKA-mediated phosphorylation of kemptide at 100 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228838(CHEMBL428973)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50358686(CHEMBL1922138)
Affinity DataIC50:  1.51E+3nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50614312(CHEMBL5284365)
Affinity DataIC50:  1.52E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50614314(CHEMBL5269818)
Affinity DataIC50:  1.53E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50597471(CHEMBL5176687)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50011236(CHEMBL344314 | Isoquinoline-5-sulfonic acid (2-ami...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228841(CHEMBL351282)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026615(CHEMBL1922045)
Affinity DataIC50:  3.34E+3nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50614313(CHEMBL5283378)
Affinity DataIC50:  3.34E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50216682(1-(5-Isoquinolinesulfonyl)-2-methylpiperazine | 1-...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM14027(5-(1,4-diazepan-1-ylsulfonyl)isoquinoline | 5-(1,4...)
Affinity DataIC50:  4.58E+3nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM14027(5-(1,4-diazepan-1-ylsulfonyl)isoquinoline | 5-(1,4...)
Affinity DataIC50:  4.58E+3nMAssay Description:In vitro inhibition of angiotensin I converting enzyme in rabbit lung with hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM15203(5-(piperazine-1-sulfonyl)isoquinoline | CHEMBL7577...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50358469(CHEMBL1922026)
Affinity DataIC50:  6.74E+3nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50206006(7,8-Dihydroxy-2H-1-benzopyran-2-one | 7,8-dihydrox...)
Affinity DataIC50:  9.33E+3nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50593027(CHEMBL5186340)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50525707(CHEMBL4457566)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PKAcgamma using [KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK] as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50431132(CHEMBL2332080)
Affinity DataIC50: >2.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50614311(CHEMBL5267373)
Affinity DataIC50: >2.00E+4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50614307(CHEMBL5278333)
Affinity DataIC50: >2.00E+4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM2581(3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^...)
Affinity DataIC50:  2.57E+4nMAssay Description:Inhibition of protein kinase AMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50054426(7-hydroxy-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of protein kinase AMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50587768(CHEMBL5172395)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM2672(3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of protein kinase AMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50228845(CHEMBL410778)
Affinity DataIC50: >7.50E+4nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228844(CHEMBL263188)
Affinity DataIC50: >7.50E+4nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228842(CHEMBL437640)
Affinity DataIC50: >7.50E+4nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50469778(CHEMBL116963)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein kinase AMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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