TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 780nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 2.06E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 2.36E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 3.87E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair