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Found 45 of ic50 for UniProtKB: P48056
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473314(CHEMBL553068)
Affinity DataIC50:  51nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50081891((R)-1-[2-(3,3-Diphenyl-propoxy)-ethyl]-piperidine-...)
Affinity DataIC50:  55nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473316(CHEMBL545694)
Affinity DataIC50:  68nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473312(CHEMBL543108)
Affinity DataIC50:  74nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50080346((R)-1-(2-Benzhydrylideneaminooxy-ethyl)-piperidine...)
Affinity DataIC50:  82nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50081888((R)-1-[2-(2-Diphenylamino-ethoxy)-ethyl]-piperidin...)
Affinity DataIC50:  90nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473321(CHEMBL563076)
Affinity DataIC50:  105nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50437146(CHEMBL1189315)
Affinity DataIC50:  184nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473306(CHEMBL556178)
Affinity DataIC50:  248nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473319(CHEMBL555856)
Affinity DataIC50:  265nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50437144(CHEMBL1190271)
Affinity DataIC50:  308nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50003634(1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxyli...)
Affinity DataIC50:  330nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473315(CHEMBL541561)
Affinity DataIC50:  460nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473313(CHEMBL545690)
Affinity DataIC50:  561nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473311(CHEMBL543342)
Affinity DataIC50:  644nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50437145(CHEMBL1196076)
Affinity DataIC50:  647nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473317(CHEMBL553053)
Affinity DataIC50:  696nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473320(CHEMBL545452)
Affinity DataIC50:  770nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473309(CHEMBL552675)
Affinity DataIC50:  851nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473302(CHEMBL555631)
Affinity DataIC50:  1.16E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473303(CHEMBL542641)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50003653(1-(2-Benzhydryloxy-ethyl)-piperidine-3-carboxylic ...)
Affinity DataIC50:  1.37E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50226144(2,4-Diamino-Butyric Acid | CHEBI:64307 | CHEMBL307...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50078167(CHEMBL69064)
Affinity DataIC50:  2.02E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473308(CHEMBL541821)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473305(CHEMBL71789)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473318(CHEMBL539773)
Affinity DataIC50:  5.51E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50003624((RS)-nipecotic acid | CHEMBL277498 | Nipecotic | P...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50223874(CHEMBL277372)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473310(CHEMBL303402)
Affinity DataIC50:  1.36E+4nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473307(CHEMBL545692)
Affinity DataIC50:  1.46E+4nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50473304(CHEMBL541556)
Affinity DataIC50: >4.00E+4nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50226141(CHEMBL309688)
Affinity DataIC50:  1.30E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50226145(CHEMBL150830)
Affinity DataIC50:  1.60E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50223872(CHEMBL15851)
Affinity DataIC50:  1.73E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50223876(CHEMBL16226)
Affinity DataIC50:  2.03E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50223871(CHEMBL429974)
Affinity DataIC50:  2.40E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50224808(CHEMBL309689)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50226143(CHEMBL305673)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50226142(CHEMBL292757)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50000106(4-CARBOXYPIPERIDINE | CHEMBL279998 | Piperidine-4-...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50223875(CHEMBL280511)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50226146(CHEMBL74364)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50223873(CHEMBL16357)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Rattus norvegicus)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50223877(CHEMBL16132)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed