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Found 6 of ki for UniProtKB: P31424
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Rattus norvegicus (Rat))
Hoffmann-La Roche

US Patent
LigandPNGBDBM143695(US9682959, 3 | US9751856, 3)
Affinity DataKi:  16nMAssay Description:The pharmacological activity of the compounds was tested using the following method: cDNA encoding rat mGlu 5a receptor was transiently transfected i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Rattus norvegicus (Rat))
Hoffmann-La Roche

US Patent
LigandPNGBDBM143693(US9682959, 1 | US9751856, 1)
Affinity DataKi:  18nMAssay Description:The pharmacological activity of the compounds was tested using the following method: cDNA encoding rat mGlu 5a receptor was transiently transfected i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Rattus norvegicus (Rat))
Hoffmann-La Roche

US Patent
LigandPNGBDBM143694(US9682959, 2 | US9751856, 2)
Affinity DataKi:  38nMAssay Description:The pharmacological activity of the compounds was tested using the following method: cDNA encoding rat mGlu 5a receptor was transiently transfected i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Rattus norvegicus (Rat))
Hoffmann-La Roche

US Patent
LigandPNGBDBM143697(US9682959, 4 | US9751856, 4)
Affinity DataKi:  80nMAssay Description:The pharmacological activity of the compounds was tested using the following method: cDNA encoding rat mGlu 5a receptor was transiently transfected i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Rattus norvegicus (Rat))
Hoffmann-La Roche

US Patent
LigandPNGBDBM143699(US9682959, 6 | US9751856, 6)
Affinity DataKi:  280nMAssay Description:The pharmacological activity of the compounds was tested using the following method: cDNA encoding rat mGlu 5a receptor was transiently transfected i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIsoform 1 of Metabotropic glutamate receptor 5 (5a)(Rattus norvegicus (Rat))
Hoffmann-La Roche

US Patent
LigandPNGBDBM143698(US9682959, 5 | US9751856, 5)
Affinity DataKi:  281nMAssay Description:The pharmacological activity of the compounds was tested using the following method: cDNA encoding rat mGlu 5a receptor was transiently transfected i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent