Compile Data Set for Download or QSAR
maximum 50k data
Found 273 of ic50 for UniProtKB: P24723
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  0.251nMAssay Description:Inhibition of human PKCeta using ERMRPRKRQGSVRRRV as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3183(2-({2,6-dihydroxy-4-[({2-[(4-hydroxybenzene)amido]...)
Affinity DataIC50:  0.600nMpH: 7.5 T: 2°CAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3153(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxybenzen...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of Protein Kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3153(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxybenzen...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3153(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxybenzen...)
Affinity DataIC50:  0.600nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3153(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxybenzen...)
Affinity DataIC50:  0.600nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50393218(CHEMBL1996510)
Affinity DataIC50:  1nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3153(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxybenzen...)
Affinity DataIC50:  1nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50285250(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  1nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3153(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxybenzen...)
Affinity DataIC50:  1nMAssay Description:Inhibition of protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3153(2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxybenzen...)
Affinity DataIC50:  1nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human PKCeta using ERMRPRKRQGSVRRRV as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50393214(CHEMBL2151411)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50393228(CHEMBL2153750)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50285240(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human Protein Kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50285239(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human Protein Kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50391897(CHEMBL2147537)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant human PKCeta assessed as [33P]-ATP incorporation into tridecapeptide substrate after 60 mins by scintillation proximity ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50055672(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  2nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50055668(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50055677(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50055685(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3149(2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(4-hydroxybenzen...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3149(2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(4-hydroxybenzen...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Protein kinase C beta 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3199((+-)-anti-2-[[2,6-Dihydroxy-4-[[[2-(4-hydroxybenzy...)
Affinity DataIC50:  3nMAssay Description:Inhibition of protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3186((S)-2-[[2,6-Dihydroxy-4-[[[3-(4-hydroxyphenyl)-2-[...)
Affinity DataIC50:  3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3149(2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(4-hydroxybenzen...)
Affinity DataIC50:  3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3199((+-)-anti-2-[[2,6-Dihydroxy-4-[[[2-(4-hydroxybenzy...)
Affinity DataIC50:  3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3149(2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(4-hydroxybenzen...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Protein kinase C zetaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50285087((R)-2-{2,6-Dihydroxy-4-[(3R,4R)-4-(4-hydroxy-benzo...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50285241(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human Protein Kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50285242(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human Protein Kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50366386(CHEMBL1794808)
Affinity DataIC50:  3nMAssay Description:Inhibition of human Protein Kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3199((+-)-anti-2-[[2,6-Dihydroxy-4-[[[2-(4-hydroxybenzy...)
Affinity DataIC50:  3nMAssay Description:Inhibition of protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3149(2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(4-hydroxybenzen...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50055684(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50393219(CHEMBL2151415)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50055676(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  4nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  4nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50391902(CHEMBL2147542)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human PKCeta assessed as [33P]-ATP incorporation into tridecapeptide substrate after 60 mins by scintillation proximity ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50285251(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3149(2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(4-hydroxybenzen...)
Affinity DataIC50:  4nMAssay Description:Inhibition of PKCeta (unknown origin) by IMAP kinase assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  4nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3248((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50:  4nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3252((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50:  4nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50285237(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human Protein Kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Protein Kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  4nMAssay Description:Inhibition of protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C eta type(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50:  4nMAssay Description:Inhibition of protein kinase C etaMore data for this Ligand-Target Pair
In DepthDetails Article
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