Affinity DataKd: 0.850nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKd: 0.850nMAssay Description:Binding constant for EPHA2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.850nMAssay Description:Binding constant for EPHA2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.80nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 3.60nMAssay Description:Binding constant for EPHA2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3.80nMAssay Description:Binding constant for EPHA2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 6.90nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 8nMAssay Description:Binding affinity to human EPHA2More data for this Ligand-Target Pair
Affinity DataKd: 9nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Inhibition of EPHA2 in human HEK293 cells after 1 hr by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Binding constant for EPHA2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 21nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 22nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 24nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 30nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 44nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 46nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 52nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 65nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 78nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 81nMAssay Description:Binding affinity to recombinant human GST-tagged EphA2 cytoplasmic domain (560 to 976 residues) expressed in baculovirus expression system by fluores...More data for this Ligand-Target Pair
Affinity DataKd: 87nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 87nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 93nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 99nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding constant for EPHA2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 107nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 115nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding constant for EPHA2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 146nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 152nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 158nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Binding constant for EPHA2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Binding constant for EPHA2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 165nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 173nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 187nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 187nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 192nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 198nMAssay Description:Kinobeads competition assays were performed in 96-well format as previously described using mixed protein lysates of four cancer cell lines (K-562, M...More data for this Ligand-Target Pair
Affinity DataKd: 202nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 204nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 230nMAssay Description:Binding constant for EPHA2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 238nMAssay Description:Inhibition of EPHA2 (unknown origin) by ITCMore data for this Ligand-Target Pair
