Affinity DataKi: 15nMAssay Description:Relative potency against Histamine H1 receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Apparent pA2 value of compound at 50 nM concentration of mepyramine in rat aortaMore data for this Ligand-Target Pair
Affinity DataKi: 2.41E+3nMAssay Description:Apparent pA2 value of compound at 10 nM concentration of mepyramine in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKi: 3.12E+3nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
Affinity DataKi: 3.80E+3nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
TargetAdenomatous polyposis coli protein [1477-1519]/Catenin beta-1 [138-686](Homo sapiens (Human))
University of Utah Research Foundation
US Patent
University of Utah Research Foundation
US Patent
Affinity DataKi: 8.31E+3nM ΔG°: -6.93kcal/molepH: 7.4 T: 2°CAssay Description:Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (...More data for this Ligand-Target Pair
Affinity DataKi: 4.46E+4nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.46E+4nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
TargetAdenomatous polyposis coli protein [1477-1519]/Catenin beta-1 [138-686](Homo sapiens (Human))
University of Utah Research Foundation
US Patent
University of Utah Research Foundation
US Patent
Affinity DataKi: 5.39E+4nM ΔG°: -5.82kcal/moleT: 2°CAssay Description:Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino...More data for this Ligand-Target Pair
TargetAdenomatous polyposis coli protein [1477-1519]/Catenin beta-1 [138-686](Homo sapiens (Human))
University of Utah Research Foundation
US Patent
University of Utah Research Foundation
US Patent
Affinity DataKi: 6.25E+4nM ΔG°: -5.73kcal/moleT: 2°CAssay Description:Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino...More data for this Ligand-Target Pair
TargetAdenomatous polyposis coli protein [1477-1519]/Catenin beta-1 [138-686](Homo sapiens (Human))
University of Utah Research Foundation
US Patent
University of Utah Research Foundation
US Patent
Affinity DataKi: 6.62E+4nM ΔG°: -5.70kcal/molepH: 7.4 T: 2°CAssay Description:Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (...More data for this Ligand-Target Pair
TargetAdenomatous polyposis coli protein [1477-1519]/Catenin beta-1 [138-686](Homo sapiens (Human))
University of Utah Research Foundation
US Patent
University of Utah Research Foundation
US Patent
Affinity DataKi: 1.71E+5nM ΔG°: -5.14kcal/molepH: 7.4 T: 2°CAssay Description:Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (...More data for this Ligand-Target Pair
TargetAdenomatous polyposis coli protein [1477-1519]/Catenin beta-1 [138-686](Homo sapiens (Human))
University of Utah Research Foundation
US Patent
University of Utah Research Foundation
US Patent
Affinity DataKi: 1.71E+5nM ΔG°: -5.13kcal/moleT: 2°CAssay Description:Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino...More data for this Ligand-Target Pair
TargetAdenomatous polyposis coli protein [1477-1519]/Catenin beta-1 [138-686](Homo sapiens (Human))
University of Utah Research Foundation
US Patent
University of Utah Research Foundation
US Patent
Affinity DataKi: 1.76E+5nM ΔG°: -5.12kcal/moleT: 2°CAssay Description:Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino...More data for this Ligand-Target Pair
