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Found 17 of ic50 for UniProtKB: P53041
TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50061067(15-(3-Guanidino-propyl)-8-isobutyl-18-((1E,3E)-6-m...)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at NK2 receptor in human urinary bladder assessed as inhibition of [beta-Ala8]NKA(4-10)-induced tissue contractionsMore data for this Ligand-Target Pair
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TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50110690(CHEMBL17377 | FOSTRIECIN | Phosphoric acid mono-{3...)
Affinity DataIC50: >1nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
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TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50110681(CHEMBL430266 | Calyculin-A)
Affinity DataIC50:  3nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
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TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50408820(CHEMBL5268133)
Affinity DataIC50:  3.5nMAssay Description:Antagonist activity at mouse histamine H4 receptor in SK-N-MC cells assessed as inhibition of forskolin-stimulated cAMP release preincubated for 10 m...More data for this Ligand-Target Pair
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TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50408822(CHEMBL5276260)
Affinity DataIC50:  4nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
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TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50366883(TAUTOMYCIN)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at mouse histamine H4 receptor in SK-N-MC cells assessed as inhibition of forskolin-stimulated cAMP release preincubated for 10 m...More data for this Ligand-Target Pair
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TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50408823(CHEMBL5276593)
Affinity DataIC50:  12nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
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TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50090505((1R,2S,6R,7S)-2,6-Dimethyl-4,10-dioxa-tricyclo[5.2...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50090505((1R,2S,6R,7S)-2,6-Dimethyl-4,10-dioxa-tricyclo[5.2...)
Affinity DataIC50:  600nMAssay Description:Antagonist activity at rat H3 receptor expressed in human SK-N-MC cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrsMore data for this Ligand-Target Pair
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TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50607111(CHEMBL5218807)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PP5 (unknown origin)More data for this Ligand-Target Pair
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TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50112358(CHEMBL3609374)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of phosphatase activity of human PP5 using pNPP as a substrate after 10 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50112357(CHEMBL3609375)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of phosphatase activity of human PP5 using pNPP as a substrate after 10 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50112356(CHEMBL3609373)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of phosphatase activity of human PP5 using pNPP as a substrate after 10 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50087856(CHEMBL3426913)
Affinity DataIC50: >5.00E+4nMpH: 7.0Assay Description:Inhibition of PP5 (unknown origin) using pNPP as substrate at pH 7 at 25 degC by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50607110(CHEMBL5219519)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PP5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50420258(CEFSULODIN)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of phosphatase activity of human PP5 using pNPP as a substrate after 10 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50558488(CHEMBL4794972)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of PP5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed