TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University
Stockholm University
Affinity DataKd: 43nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
Affinity DataKd: 26nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells incubated for 60 mins in presence of NT (8 to 13) without compound was...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University
Stockholm University
Affinity DataKd: 1.20E+3nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University
Stockholm University
Affinity DataKd: 1.60E+3nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University
Stockholm University
Affinity DataKd: 2.10E+3nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University
Stockholm University
Affinity DataKd: 1.80E+4nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University
Stockholm University
Affinity DataKd: 4.20E+4nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University
Stockholm University
Affinity DataKd: 1.00E+3nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University
Stockholm University
Affinity DataKd: 2.80E+3nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University
Stockholm University
Affinity DataKd: 1.90E+3nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University
Stockholm University
Affinity DataKd: 1.76E+4nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University
Stockholm University
Affinity DataKd: 4.15E+4nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
Affinity DataKd: 1.55nMAssay Description:Binding affinity to human recombinant NTS1 in HEK293T cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding affinity to human recombinant NTS1 in HEK293T cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.510nMAssay Description:Binding affinity to NTSR1 in human HT-29 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKd: 0.440nMAssay Description:Binding affinity to NTSR1 in human HT-29 cells after 2 hrs by liquid scintillation counting in presence of NTSR2 ligand (S)-2-((2S,3S)-2-(2-((S)-1-((...More data for this Ligand-Target Pair
Affinity DataKd: 0.580nMAssay Description:Binding affinity to human NTSR1 receptor transfected in CHO cells co-expressing Galpha16-mtAEQ after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKd: 0.590nMAssay Description:Displacement of [3H]neurotensin from human NTS1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.160nMAssay Description:In vitro inhibition of [3H]-NT binding to human striatal Neurotensin receptor 1More data for this Ligand-Target Pair
Affinity DataKd: 0.510nMAssay Description:Displacement of [3H]neurotensin from human NTS1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.630nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 8.90nMAssay Description:Displacement of [3H]SR48692 from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKd: 2.5nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells incubated for 75 mins in presence of NT (8 to 13) followed by compound...More data for this Ligand-Target Pair
Affinity DataKd: 3.60nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells preincubated for 20 mins to 2 hrs followed by addition of NT (8 to 13)...More data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells incubated for 60 mins in presence of NT (8 to 13) without compound was...More data for this Ligand-Target Pair
Affinity DataKd: 6.30nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells incubated for 60 mins in presence of NT (8 to 13) without compound was...More data for this Ligand-Target Pair
Affinity DataKd: 8.10nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells incubated for 75 mins in presence of NT (8 to 13) followed by compound...More data for this Ligand-Target Pair
Affinity DataKd: 3.80nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells incubated for 75 mins in presence of NT (8 to 13) followed by compound...More data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells incubated for 60 mins in presence of NT (8 to 13) without compound was...More data for this Ligand-Target Pair
Affinity DataKd: 6.80nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells incubated for 75 mins in presence of NT (8 to 13) followed by compound...More data for this Ligand-Target Pair
Affinity DataKd: 3.90nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells preincubated for 20 mins to 2 hrs followed by addition of NT (8 to 13)...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University
Stockholm University
Affinity DataKd: 0.400nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
