Affinity DataKi: 12.5nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 12.7nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 15.3nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity towards Lysophosphatidic acid 1 (LPA1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:In vitro ability to antagonize LPA-evoked [35S]-GTP-gammaS binding to lysophosphatidic acid receptor 1 in HEK293T cell linesMore data for this Ligand-Target Pair
Affinity DataKi: 18.8nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity towards Lysophosphatidic acid 1 (LPA1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24.5nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity towards Lysophosphatidic acid 1 (LPA1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 27.6nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity towards Lysophosphatidic acid 1 (LPA1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 30.8nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:In vitro ability to antagonize LPA-evoked [35S]-GTP-gammaS binding to lysophosphatidic acid receptor 1 in HEK293T cell linesMore data for this Ligand-Target Pair
Affinity DataKi: 34.6nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Binding affinity towards Lysophosphatidic acid 1 (LPA1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 40.9nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 44.2nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 46.2nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity to LPA1More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Antagonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
Affinity DataKi: 51.4nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 53.8nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 60.7nMAssay Description:Activity at human LPA1 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Binding affinity towards Lysophosphatidic acid 1 (LPA1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 72.3nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:In vitro ability to antagonize LPA-evoked [35S]-GTP-gammaS binding to lysophosphatidic acid receptor 1 in HEK293T cell linesMore data for this Ligand-Target Pair
Affinity DataKi: 80.5nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Competitive antagonist activity at human LPA1 receptor overexpressed in CHO cells assessed as inhibition of LPA-induced [35S]GTPgammaS binding by liq...More data for this Ligand-Target Pair
Affinity DataKi: 94.8nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:The ability of a compound to inhibit binding of a ligand (1-(4′-(4-(((benzyloxy)carbonyl)amino)-3-methylisoxazol-5-yl)-[1,1′-biphenyl]-4-...More data for this Ligand-Target Pair
Affinity DataKi: 134nMAssay Description:In vitro ability to antagonize LPA-evoked [35S]-GTP-gammaS binding to lysophosphatidic acid receptor 1 in HEK293T cell linesMore data for this Ligand-Target Pair
Affinity DataKi: 137nMAssay Description:In vitro ability to antagonize LPA-evoked [35S]-GTP-gammaS binding to lysophosphatidic acid receptor 1 in HEK293T cell linesMore data for this Ligand-Target Pair
Affinity DataKi: 139nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 143nMAssay Description:Competitive antagonist activity at human LPA1 receptor overexpressed in CHO cells assessed as inhibition of LPA-induced [35S]GTPgammaS binding by liq...More data for this Ligand-Target Pair
Affinity DataKi: 156nMAssay Description:In vitro ability to antagonize LPA-evoked [35S]-GTP-gammaS binding to lysophosphatidic acid receptor 1 in HEK293T cell linesMore data for this Ligand-Target Pair
Affinity DataKi: 156nMAssay Description:Binding affinity towards Lysophosphatidic acid 1 (LPA1) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 221nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 311nMAssay Description:Binding affinity to LPA1More data for this Ligand-Target Pair
Affinity DataKi: 314nMAssay Description:Activity at human LPA1 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataKi: 358nMAssay Description:In vitro ability to antagonize LPA-evoked [35S]-GTP-gammaS binding to lysophosphatidic acid receptor 1 in HEK293T cell linesMore data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 403nMAssay Description:Activity at human LPA1 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataKi: 407nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 425nMAssay Description:Binding affinity for Lysophosphatidic acid receptor 1 expressed in RH7777 rat hepatoma cellsMore data for this Ligand-Target Pair
Affinity DataKi: 457nMAssay Description:Binding affinity for Lysophosphatidic acid receptor 1 expressed in RH7777 rat hepatoma cellsMore data for this Ligand-Target Pair
Affinity DataKi: 788nMAssay Description:Binding affinity for Lysophosphatidic acid receptor 1 expressed in RH7777 rat hepatoma cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.08E+3nMAssay Description:Binding affinity for Lysophosphatidic acid receptor 1 expressed in RH7777 rat hepatoma cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.15E+3nMAssay Description:Binding affinity for Lysophosphatidic acid receptor 1 expressed in RH7777 rat hepatoma cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.35E+3nMAssay Description:Binding affinity for Lysophosphatidic acid receptor 1 expressed in RH7777 rat hepatoma cellsMore data for this Ligand-Target Pair