TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK2/Cyclin E expressed in baculovirus infected Sf9 cells using histone H1 substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human full length N-terminal GST-HIS6 fused CDK9 (M1 to F372 residues)/N-terminal HIS6-fused Cyclin-T1 (M1 to K726 residues) co-express...More data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human full length N-terminal GST-HIS6 fused CDK9 (M1 to F372 residues)/N-terminal HIS6-fused Cyclin-T1 (M1 to K726 residues) co-express...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Egyptian Russian University
Curated by ChEMBL
Egyptian Russian University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK2/Cyclin E expressed in baculovirus infected Sf9 cells using histone H1 substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair