Affinity DataKi: 0.0500nMAssay Description:Binding affinity to human recombinant JAK2 assessed as inhibition constant incubated for 30 mins by microtiter plate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Binding affinity to human recombinant JAK1 assessed as inhibition constant incubated for 30 mins by microtiter plate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human recombinant CRF1 in HEK cell line assessed as inhibition constant incubated for 2 hrs by MicroBeta scintillation counter me...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to A beta-amyloid plaque (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.69E+4nMAssay Description:Binding affinity to human recombinant CRF2 in HEK cell line assessed as inhibition constant incubated for 4 to 5 hrs by Scintillation Proximity AssayMore data for this Ligand-Target Pair