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TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))TBA
LigandPNGBDBM50609298(CHEMBL5268404)
Affinity DataKi:  0.0500nMAssay Description:Binding affinity to human recombinant JAK2 assessed as inhibition constant incubated for 30 mins by microtiter plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))TBA
LigandPNGBDBM50609298(CHEMBL5268404)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to human recombinant JAK1 assessed as inhibition constant incubated for 30 mins by microtiter plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50272695(3-(4-chloro-2-morpholinothiazol-5-yl)-2,6-dimethyl...)
Affinity DataKi:  10nMAssay Description:Binding affinity to human recombinant CRF1 in HEK cell line assessed as inhibition constant incubated for 2 hrs by MicroBeta scintillation counter me...More data for this Ligand-Target Pair
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TargetAmyloid-beta precursor protein(Homo sapiens (Human))TBA
LigandPNGBDBM50122787(2-(4'-dimethylaminophenyl)-6-iodoimidazo[1,2-a]pyr...)
Affinity DataKi:  11nMAssay Description:Binding affinity to A beta-amyloid plaque (unknown origin)More data for this Ligand-Target Pair
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TargetCorticotropin-releasing factor receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50272695(3-(4-chloro-2-morpholinothiazol-5-yl)-2,6-dimethyl...)
Affinity DataKi:  1.69E+4nMAssay Description:Binding affinity to human recombinant CRF2 in HEK cell line assessed as inhibition constant incubated for 4 to 5 hrs by Scintillation Proximity AssayMore data for this Ligand-Target Pair
In DepthDetails PubMed