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Found 24 Enz. Inhib. hit(s) with all data for entry = 11722
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642632(US20230416245, Compound 70)
Affinity DataKi:  0.133nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642621(US20230416245, Compound 59)
Affinity DataKi:  0.230nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642624(US20230416245, Compound 62)
Affinity DataKi:  0.330nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642626(US20230416245, Compound 64)
Affinity DataKi:  0.640nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642625(US20230416245, Compound 63)
Affinity DataKi:  0.720nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642618(US20230416245, Compound 45)
Affinity DataKi:  1.30nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642635(US20230416245, Compound 83)
Affinity DataKi:  1.62nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642631(US20230416245, Compound 69)
Affinity DataKi:  1.68nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642620(US20230416245, Compound 35)
Affinity DataKi:  1.70nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642615(US20230416245, Compound 40)
Affinity DataKi:  2nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642636(US20230416245, Compound 90)
Affinity DataKi:  2.42nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642639(US20230416245, Compound 93)
Affinity DataKi:  2.59nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642627(US20230416245, Compound 65)
Affinity DataKi:  3.49nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642630(US20230416245, Compound 68)
Affinity DataKi:  4.75nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642634(US20230416245, Compound 82)
Affinity DataKi:  4.77nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642637(US20230416245, Compound 91)
Affinity DataKi:  5.10nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642623(US20230416245, Compound 61)
Affinity DataKi:  7.15nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642619(US20230416245, Compound 46)
Affinity DataKi:  21.3nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642638(US20230416245, Compound 92)
Affinity DataKi:  26.8nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642617(US20230416245, Compound 44)
Affinity DataKi:  28.4nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642629(US20230416245, Compound 67)
Affinity DataKi:  94.4nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642628(US20230416245, Compound 66)
Affinity DataKi:  126nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642633(US20230416245, Compound 71)
Affinity DataKi:  456nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A3(Homo sapiens (Human))
Biointervene

US Patent
LigandPNGBDBM642622(US20230416245, Compound 60)
Affinity DataKi: >9.40E+3nMAssay Description:Radioligand-binding assays were performed using the adenosine A3 receptor agonist [125I]-AB-MECA and the A1 receptor agonist [3H]CCPA. Binding assays...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent