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Found 15 Enz. Inhib. hit(s) with all data for entry = 5047
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50005836(4-Amino-5-chloro-N-{1-[3-(4-fluoro-phenoxy)-propyl...)
Affinity DataKi:  25nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82422(CAS_109872-41-5 | NSC_3035240 | RENZAPRIDE)
Affinity DataKi:  27nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82087(2-(5-methoxy-1H-indol-3-yl)ethanamine | 5-MT | 5-M...)
Affinity DataKi:  112nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50005836(4-Amino-5-chloro-N-{1-[3-(4-fluoro-phenoxy)-propyl...)
Affinity DataKi:  122nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50000492((zacopride)4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataKi:  136nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi:  145nMMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50007871(CHEMBL8197 | ICS 205-930 | TROPISETRON)
Affinity DataKi:  159nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82422(CAS_109872-41-5 | NSC_3035240 | RENZAPRIDE)
Affinity DataKi:  243nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM81781(5-HT,a-Me | 5-HT,omega-N-Me)
Affinity DataKi:  263nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82087(2-(5-methoxy-1H-indol-3-yl)ethanamine | 5-MT | 5-M...)
Affinity DataKi:  401nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50007871(CHEMBL8197 | ICS 205-930 | TROPISETRON)
Affinity DataKi:  544nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50000492((zacopride)4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataKi:  808nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM21392(3-(2-aminoethyl)-1H-indole-5-carboxamide | 5-CT | ...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM81781(5-HT,a-Me | 5-HT,omega-N-Me)
Affinity DataKi:  1.45E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed