Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50035611
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM18134(({[({[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibitory constant against rat Methionine adenosyltransferase was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM18134(({[({[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-...)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367305(CHEMBL1791430)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibitory constant against rat liver Methionine adenosyltransferase I, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367303(CHEMBL1791433)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibitory constant against rat liver Methionine adenosyltransferase I, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367042(CHEMBL606221)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibitory constant against rat liver Methionine adenosyltransferase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367301(CHEMBL1791432)
Affinity DataKi:  3.70E+4nMAssay Description:Competitive inhibition of rat methionine adenosyltransferase, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367301(CHEMBL1791432)
Affinity DataKi:  4.80E+4nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase II, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367042(CHEMBL606221)
Affinity DataKi:  7.50E+4nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367305(CHEMBL1791430)
Affinity DataKi:  8.00E+4nMAssay Description:Competitive inhibition of rat methionine adenosyltransferase, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367300(CHEMBL610977)
Affinity DataKi:  1.00E+5nMAssay Description:Competitive inhibition of rat methionine adenosyltransferase, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
Affinity DataKi:  1.10E+5nMAssay Description:Inhibitory constant against rat Methionine adenosyltransferase was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026197(Adenosine 5'-triphosphate derivative | CHEMBL31428...)
Affinity DataKi:  1.40E+5nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase II, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367307(CHEMBL1791431)
Affinity DataKi:  1.40E+5nMAssay Description:Competitive inhibition of rat methionine adenosyltransferase, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026193(Adenosine 5'-triphosphate derivative | CHEMBL31428...)
Affinity DataKi:  1.70E+5nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase II, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026197(Adenosine 5'-triphosphate derivative | CHEMBL31428...)
Affinity DataKi:  1.70E+5nMAssay Description:Competitive inhibition of rat methionine adenosyltransferase, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026193(Adenosine 5'-triphosphate derivative | CHEMBL31428...)
Affinity DataKi:  1.80E+5nMAssay Description:Competitive inhibition of rat methionine adenosyltransferase, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367305(CHEMBL1791430)
Affinity DataKi:  1.90E+5nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase II, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367304(CHEMBL610404)
Affinity DataKi:  2.10E+5nMAssay Description:Inhibitory constant against rat methionine adenosyltransferase was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367307(CHEMBL1791431)
Affinity DataKi:  2.70E+5nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase II, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50118221(9H-purine derivative | CHEMBL132722 | DIPHOSPHOMET...)
Affinity DataKi:  3.00E+5nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367300(CHEMBL610977)
Affinity DataKi:  3.10E+5nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase II, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367042(CHEMBL606221)
Affinity DataKi:  3.10E+5nMAssay Description:Inhibitory constant against rat Methionine adenosyltransferase was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50118221(9H-purine derivative | CHEMBL132722 | DIPHOSPHOMET...)
Affinity DataKi:  3.40E+5nMAssay Description:Inhibitory constant against rat Methionine adenosyltransferase was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367303(CHEMBL1791433)
Affinity DataKi:  4.10E+5nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase II, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367306(CHEMBL608929)
Affinity DataKi:  5.20E+5nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50010308(CHEMBL3251357)
Affinity DataKi:  5.30E+5nMAssay Description:Inhibitory constant against rat Methionine adenosyltransferase was reportedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367304(CHEMBL610404)
Affinity DataKi:  5.30E+5nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
Affinity DataKi:  6.00E+5nMAssay Description:Inhibitory constant against rat kidney Methionine adenosyltransferase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1/type-2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367303(CHEMBL1791433)
Affinity DataKi:  7.50E+5nMAssay Description:Competitive inhibition of rat methionine adenosyltransferase, activity expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-adenosylmethionine synthase isoform type-1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367306(CHEMBL608929)
Affinity DataKi:  3.30E+6nMAssay Description:Inhibitory constant against rat liver Methionine adenosyltransferase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed