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Found 27 Enz. Inhib. hit(s) with all data for entry = 50010827
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099151(CHEMBL177442 | N'-[5-(4-{4-[(S)-2-Hydroxy-3-(2-oxo...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of 125 I-Iodocyanopindolol binding to Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099151(CHEMBL177442 | N'-[5-(4-{4-[(S)-2-Hydroxy-3-(2-oxo...)
Affinity DataKi:  7.20nMAssay Description:Inhibition of 125 I-Iodocyanopindolol binding to Beta-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099160(CHEMBL354906 | [5-(4-{4-[(R)-2-Hydroxy-2-(4-hydrox...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of 125 I-Iodocyanopindolol binding to Beta-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099160(CHEMBL354906 | [5-(4-{4-[(R)-2-Hydroxy-2-(4-hydrox...)
Affinity DataKi:  9.10E+3nMAssay Description:Inhibition of 125 I-Iodocyanopindolol binding to Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099150(CHEMBL368584 | N-[5-(2-{1-[4-((R)-3,5-Dioxo-[1,2,4...)
Affinity DataKi:  9.49E+3nMAssay Description:Inhibition of 125 I-Iodocyanopindolol binding to Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099150(CHEMBL368584 | N-[5-(2-{1-[4-((R)-3,5-Dioxo-[1,2,4...)
Affinity DataKi:  7.40E+4nMAssay Description:Inhibition of 125 I-Iodocyanopindolol binding to Beta-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099155(CHEMBL174054 | N-[2-Hydroxy-5-(1-hydroxy-2-{1-[4-(...)
Affinity DataEC50:  34nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099156(CHEMBL174534 | N'-(5-{4-[4-((S)-2-Hydroxy-3-phenox...)
Affinity DataEC50:  940nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099157(CHEMBL435307 | N-[2-Hydroxy-5-((S)-2-hydroxy-3-{1-...)
Affinity DataEC50:  1nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099166(CHEMBL367561 | N'-[5-(4-{4-[(S)-2-Hydroxy-3-(8-hyd...)
Affinity DataEC50:  2nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099158(4-((S)-2-Hydroxy-3-{1-[4-(4-oxo-2-piperidin-1-yl-4...)
Affinity DataEC50:  9nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099159(CHEMBL174442 | N-[2-Hydroxy-5-((R)-1-hydroxy-2-{1-...)
Affinity DataEC50:  9nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099160(CHEMBL354906 | [5-(4-{4-[(R)-2-Hydroxy-2-(4-hydrox...)
Affinity DataEC50:  34nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099161(CHEMBL177185 | N-[5-(2-{1-[4-(2,4-Dioxo-thiazolidi...)
Affinity DataEC50:  6nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099162(CHEMBL177438 | N-[2-Hydroxy-5-(1-hydroxy-2-{1-[4-(...)
Affinity DataEC50:  86nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099164(CHEMBL366657 | N-[5-((R)-2-{1-[4-(2-Cyanoamino-4-o...)
Affinity DataEC50:  10nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099165(8-Hydroxy-5-((S)-2-hydroxy-3-{1-[4-(4-oxo-2-piperi...)
Affinity DataEC50:  6nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099163(CHEMBL178848 | N-[2-Hydroxy-5-((R)-1-hydroxy-2-{1-...)
Affinity DataEC50:  80nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099167(CHEMBL369155 | N'-[5-(4-{4-[(S)-2-Hydroxy-3-(4-hyd...)
Affinity DataEC50:  400nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099168(CHEMBL177400 | N-{5-[(R)-2-(1-{4-[2-(N',N'-Dimethy...)
Affinity DataEC50:  3nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099154(CHEMBL173472 | N-[2-Hydroxy-5-(1-hydroxy-2-{1-[4-(...)
Affinity DataEC50:  9nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099153(CHEMBL451185 | N-[2-Hydroxy-5-(1-hydroxy-2-{1-[4-(...)
Affinity DataEC50:  230nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099152(CHEMBL366395 | N-{5-[(R)-2-(1-{4-[2-(1-Benzyl-pipe...)
Affinity DataEC50:  90nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099151(CHEMBL177442 | N'-[5-(4-{4-[(S)-2-Hydroxy-3-(2-oxo...)
Affinity DataEC50:  10nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099150(CHEMBL368584 | N-[5-(2-{1-[4-((R)-3,5-Dioxo-[1,2,4...)
Affinity DataEC50:  20nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099149(5-{4-[4-((S)-2-Hydroxy-3-phenoxy-propylamino)-pipe...)
Affinity DataEC50:  75nMAssay Description:Beta 3-adrenergic receptor agonistic activity, evaluated by measurement of cAMP accumulation in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50097798(CHEMBL163262 | N-[5-((R)-2-{1-[4-(2,4-Dioxo-thiazo...)
Affinity DataEC50:  10nMAssay Description:Beta 3-adrenergic receptor agonistic activity as cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed