Affinity DataKi: 0.5nMAssay Description:Binding affinity to KOR (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.597nMAssay Description:Binding affinity to KOR (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity to human cloned MOR in presence of Na+/GDPMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [3H]diprenorphine from KOR (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [3H]diprenorphine from rat cloned KOR expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Displacement of [3H]diprenorphine from rat cloned KOR expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 122nMAssay Description:Binding affinity to human cloned DOR in presence of Na+/GDPMore data for this Ligand-Target Pair
Affinity DataKi: 259nMAssay Description:Displacement of [3H]DAMGO from rat cloned MOR expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 619nMAssay Description:Displacement of [3H]DAMGO from rat cloned MOR expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.91E+3nMAssay Description:Displacement of [3H]DPDPE from mouse cloned DOR expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.15E+3nMAssay Description:Displacement of [3H]DPDPE from mouse cloned DOR expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5.88E+3nMAssay Description:Displacement of [3H]DAMGO from MOR (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPDPE from DOR (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Displacement of [3H]Cl-977 from KOR in guinea pig brain membrane fraction after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Antagonist activity at KOR (unknown origin) by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Displacement of DAGO from MOR in guinea pig brain membrane fraction after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at DOR (unknown origin) by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at MOR (unknown origin) by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair