Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50013582
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of Src protein tryrosine kinase dependent cellular proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132153((2,4-Dichloro-5-methoxy-phenyl)-[7-methoxy-8-(2-me...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132160((2,4-Dichloro-5-methoxy-phenyl)-(7,8-dimethoxy-4a,...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM4492(4-[(2,4-Dichlorophenyl)amino]-6,7-dimethoxy-3-quin...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132158((2,4-Dichloro-5-methoxy-phenyl)-[8-methoxy-7-(2-me...)
Affinity DataIC50:  9.80nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132153((2,4-Dichloro-5-methoxy-phenyl)-[7-methoxy-8-(2-me...)
Affinity DataIC50:  28nMAssay Description:Inhibition of Src protein tryrosine kinase dependent cellular proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM4525(4-Phenylamino-3-quinolinecarbonitrile deriv. 1c | ...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Src protein tryrosine kinase dependent cellular proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132154((2,4-Dichloro-phenyl)-[7-methoxy-8-(2-methoxy-etho...)
Affinity DataIC50:  120nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132154((2,4-Dichloro-phenyl)-[7-methoxy-8-(2-methoxy-etho...)
Affinity DataIC50:  120nMAssay Description:Inhibition of Src protein tryrosine kinase dependent cellular proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132158((2,4-Dichloro-5-methoxy-phenyl)-[8-methoxy-7-(2-me...)
Affinity DataIC50:  140nMAssay Description:Inhibition of Src protein tryrosine kinase dependent cellular proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132160((2,4-Dichloro-5-methoxy-phenyl)-(7,8-dimethoxy-4a,...)
Affinity DataIC50:  190nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataIC50:  410nMAssay Description:Inhibition of Fyn dependent cellular proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132155(7,8-Dimethoxy-5,10-dihydro-1H-pyrimido[4,5-b]quino...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132156((2,4-Dichloro-5-methoxy-phenyl)-(7,8-dimethoxy-pyr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132159((2,4-Dichloro-5-methoxy-phenyl)-[7-methoxy-8-(2-me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Src protein tryrosine kinase dependent cellular proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132156((2,4-Dichloro-5-methoxy-phenyl)-(7,8-dimethoxy-pyr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Src protein tryrosine kinase dependent cellular proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132153((2,4-Dichloro-5-methoxy-phenyl)-[7-methoxy-8-(2-me...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Fyn dependent cellular proliferation of rat 2 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50132157(7,8-Dimethoxy-1H-pyrimido[4,5-b]quinolin-4-one | 7...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of Src protein tryrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed