Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50045177
TargetSubstance-K receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50048413(CHEMBL2370064)
Affinity DataKi:  0.155nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50001447(CHEMBL217406 | His-Lys-Thr-Asp-Ser-Phe-Val-Gly-Leu...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50048411(CHEMBL3360196)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50048410(CHEMBL3360197)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50048409(CHEMBL3360198)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50048408(CHEMBL3360199)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50048406(CHEMBL3360201)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50048407(CHEMBL3360200)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50048405(CHEMBL3360202)
Affinity DataKi:  1.95E+3nMAssay Description:Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50048415(CHEMBL3360194)
Affinity DataIC50:  5.20nMAssay Description:Displacement of [125I]SDF1 from CXCR4 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50048414(CHEMBL3360195)
Affinity DataIC50:  6.70nMAssay Description:Displacement of [125I]SDF1 from CXCR4 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed