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Found 18 Enz. Inhib. hit(s) with all data for entry = 50045254
TargetAurora kinase B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  1nMAssay Description:Inhibition of Aurora B (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053262(CHEMBL3322935)
Affinity DataIC50:  370nMAssay Description:Inhibition of Aurora A (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053263(CHEMBL3322937)
Affinity DataIC50:  690nMAssay Description:Inhibition of Aurora A (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053269(CHEMBL3323022)
Affinity DataIC50:  720nMAssay Description:Inhibition of Aurora A (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053264(CHEMBL3322940)
Affinity DataIC50:  1.44E+3nMAssay Description:Inhibition of Aurora A (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053299(CHEMBL3323024)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of Aurora A (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053270(CHEMBL3323023)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of Aurora A (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053303(CHEMBL3321770)
Affinity DataIC50:  1.82E+3nMAssay Description:Inhibition of Aurora A (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053301(CHEMBL3323029)
Affinity DataIC50:  1.88E+3nMAssay Description:Inhibition of Aurora A (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053261(CHEMBL3322933)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibition of Aurora A (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053262(CHEMBL3322935)
Affinity DataIC50:  3.58E+3nMAssay Description:Inhibition of Aurora B (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053300(CHEMBL3323025)
Affinity DataIC50:  3.83E+3nMAssay Description:Inhibition of Aurora A (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053302(CHEMBL3323030)
Affinity DataIC50:  4.16E+3nMAssay Description:Inhibition of Aurora A (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053263(CHEMBL3322937)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of Aurora B (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053302(CHEMBL3323030)
Affinity DataIC50:  2.18E+4nMAssay Description:Inhibition of Aurora B (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053269(CHEMBL3323022)
Affinity DataIC50:  3.19E+4nMAssay Description:Inhibition of Aurora B (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053261(CHEMBL3322933)
Affinity DataIC50:  4.75E+4nMAssay Description:Inhibition of Aurora B (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50053303(CHEMBL3321770)
Affinity DataIC50:  6.32E+4nMAssay Description:Inhibition of Aurora B (unknown origin) using [33P]-ATP and 10 uM ATP after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed