Compile Data Set for Download or QSAR
maximum 50k data
Found 32 Enz. Inhib. hit(s) with all data for entry = 50021228
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222356(3-(((R)-6-(4-aminophenyl)-1-((S)-1-(4-methoxypheny...)
Affinity DataIC50:  18nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222360(Ac-Asp-Arg-Leu-Asp-Ser-OH | CHEMBL238484)
Affinity DataIC50:  25nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222359(2-{[1-(4-aminobutyl)-4-methyl-2-oxo-6-phenyl-1,2,5...)
Affinity DataIC50:  38nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222359(2-{[1-(4-aminobutyl)-4-methyl-2-oxo-6-phenyl-1,2,5...)
Affinity DataIC50:  43nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222349(2-{[(6S)-1-[(1S)-1-(4-aminophenyl)ethyl]-4-methyl-...)
Affinity DataIC50:  57nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222349(2-{[(6S)-1-[(1S)-1-(4-aminophenyl)ethyl]-4-methyl-...)
Affinity DataIC50:  71nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222361(2-({1-[(4-aminophenyl)methyl]-4-methyl-2-oxo-6-phe...)
Affinity DataIC50:  170nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222347(3-(((S)-6-(4-aminophenyl)-1-((S)-1-(4-methoxypheny...)
Affinity DataIC50:  240nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222361(2-({1-[(4-aminophenyl)methyl]-4-methyl-2-oxo-6-phe...)
Affinity DataIC50:  600nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222357(3-(((R)-1-((S)-1-(4-aminophenyl)ethyl)-4-methyl-2-...)
Affinity DataIC50:  1.51E+4nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222356(3-(((R)-6-(4-aminophenyl)-1-((S)-1-(4-methoxypheny...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222357(3-(((R)-1-((S)-1-(4-aminophenyl)ethyl)-4-methyl-2-...)
Affinity DataIC50:  3.51E+4nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222353(2-({1-[(4-aminophenyl)methyl]-4-methyl-2-oxo-6-phe...)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222351(3-((1-(4-carbamimidoylbenzyl)-4-methyl-2-oxo-6-phe...)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222360(Ac-Asp-Arg-Leu-Asp-Ser-OH | CHEMBL238484)
Affinity DataIC50:  2.59E+5nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222352(CHEMBL239333 | N-{6-(4-carbamimidoyl-phenyl)-1-[(S...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222351(3-((1-(4-carbamimidoylbenzyl)-4-methyl-2-oxo-6-phe...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222350(2-((1-(4-carbamimidoylbenzyl)-4-methyl-2-oxo-6-phe...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222358(2-({1-[(4-aminophenyl)methyl]-4-methyl-2-oxo-6-phe...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222346(2-((1-(4-carbamimidoylbenzyl)-4-methyl-2-oxo-6-phe...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222348(3-(3-(3-amino-N-propylpropanamido)-4-methyl-2-oxo-...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222350(2-((1-(4-carbamimidoylbenzyl)-4-methyl-2-oxo-6-phe...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222352(CHEMBL239333 | N-{6-(4-carbamimidoyl-phenyl)-1-[(S...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222347(3-(((S)-6-(4-aminophenyl)-1-((S)-1-(4-methoxypheny...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222346(2-((1-(4-carbamimidoylbenzyl)-4-methyl-2-oxo-6-phe...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222358(2-({1-[(4-aminophenyl)methyl]-4-methyl-2-oxo-6-phe...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222355(3-(3-(6-amino-N-propylhexanamido)-4-methyl-2-oxo-6...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222348(3-(3-(3-amino-N-propylpropanamido)-4-methyl-2-oxo-...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222354(4-((1-(4-carbamimidoylbenzyl)-4-methyl-2-oxo-6-phe...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222354(4-((1-(4-carbamimidoylbenzyl)-4-methyl-2-oxo-6-phe...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222353(2-({1-[(4-aminophenyl)methyl]-4-methyl-2-oxo-6-phe...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alpha5beta1-mediated K562 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50222355(3-(3-(6-amino-N-propylhexanamido)-4-methyl-2-oxo-6...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of integrin alphavbeta3-mediated SK-MEL-24 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed