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Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50025601
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50247550(4-(5-Bromoindole-3-yl)-6,7-dimethoxyquinazoline | ...)
Affinity DataIC50:  131nMAssay Description:Inhibition of human EGFR tyrosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50247551(4-(5-Chloro-6-fluoroindole-3-yl)-6,7-dimethoxyquin...)
Affinity DataIC50:  209nMAssay Description:Inhibition of human EGFR tyrosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50247161(4-(5-Chloro-6-fluoroindole-3-yl)-7-methoxy-6-(3-mo...)
Affinity DataIC50:  333nMAssay Description:Inhibition of human EGFR tyrosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50247160(4-(5-Chloro-6-fluoro-indole-3-yl)-6,7-di-(2-methox...)
Affinity DataIC50:  472nMAssay Description:Inhibition of human EGFR tyrosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50247159(4-(6-Fluoro-5-methylindole-3-yl)-6,7-dimethoxyquin...)
Affinity DataIC50:  533nMAssay Description:Inhibition of human EGFR tyrosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM4363((2E)-2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enethio...)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibition of human EGFR tyrosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM4363((2E)-2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enethio...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of human HER2 tyrosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed