Affinity DataKi: 30.8nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 45.2nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 133nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 134nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 167nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 325nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.38E+3nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.91E+3nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.02E+4nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.30E+4nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.84E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.01E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.22E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.01E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 7.56E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.66E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.12E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.56E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.25E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 73nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 82nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 37nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataEC50: 180nMAssay Description:Agonist activity at human recombinant alpha2A adrenergic receptor expressed in CHO cells assessed as induction of [35S]GTPgammaS binding after 60 min...More data for this Ligand-Target Pair