Compile Data Set for Download or QSAR
maximum 50k data
Found 58 Enz. Inhib. hit(s) with all data for entry = 50032850
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318595(6-Bromo-7-[4-(5-methyl-isoxazol-3-ylmethyl)-pipera...)
Affinity DataIC50:  2nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318575(2-{4-[6-Chloro-2-(4-morpholin-4-ylmethylphenyl)-3H...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50335612(3-((4-(2-(4-((1H-pyrazol-1-yl)methyl)phenyl)-6-chl...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50335617(4-(4-(6-bromo-7-(4-(pyridin-4-ylmethyl)piperazin-1...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318590(4-(4-(6-Bromo-7-(4-(pyrimidin-5-ylmethyl)piperazin...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318602(4-(4-(6-Bromo-7-(4-(thiazol-4-ylmethyl)piperazin-1...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318589(6-Bromo-2-(4-methoxyphenyl)-7-(4-(pyrimidin-5-ylme...)
Affinity DataIC50:  8nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50335615(6-bromo-2-(4-methoxyphenyl)-7-(4-(pyridin-4-ylmeth...)
Affinity DataIC50:  9nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318605((4-(6-Bromo-7-(4-((5-methylisoxazol-3-yl)methyl)pi...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318603(3-((4-(6-Bromo-2-(4-(piperazin-1-ylmethyl)phenyl)-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50335608(3-((4-(6-bromo-2-(4-(piperazin-1-yl)phenyl)-3H-imi...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50335611(3-((4-(2-(4-((1H-pyrazol-1-yl)methyl)phenyl)-6-bro...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50335610(3-((4-(6-chloro-2-(4-(4-methylpiperazin-1-yl)pheny...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318592(6-BROMO-7-[4-(4-CHLOROBENZYL)PIPERAZIN-1-YL]-2-[4-...)
Affinity DataIC50:  12nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50335607(1-(4'-(6-bromo-7-(4-((5-methylisoxazol-3-yl)methyl...)
Affinity DataIC50:  14nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50335609(3-((4-(6-bromo-2-(4-(4-methylpiperazin-1-yl)phenyl...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318572(2-{4-[6-Bromo-2-(4-dimethylaminomethylphenyl)-3H-i...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318594(6-Bromo-2-(4-methoxyphenyl)-7-[4-(5-methyl-isoxazo...)
Affinity DataIC50:  17nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318608(2-(4-(6-Chloro-7-(4-((5-methylisoxazol-3-yl)methyl...)
Affinity DataIC50:  29nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318607(2-(4-(6-Bromo-7-(4-((5-methylisoxazol-3-yl)methyl)...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318600(4-(4-(6-Bromo-7-(4-((1-methyl-1H-imidazol-2-yl)met...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318599(6-Bromo-2-(4-methoxyphenyl)-7-(4-((1-methyl-1H-imi...)
Affinity DataIC50:  32nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318591(6-Bromo-7-[4-(4-chlorobenzyl)-piperazin-1-yl]-2-(4...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50224734(2-(4-(6-Chloro-2-(4-(dimethylamino)phenyl)-3H-imid...)
Affinity DataIC50:  42nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318569(2-(4-(6-Cyano-2-(4-(dimethylamino)phenyl)-3H-imida...)
Affinity DataIC50:  50nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318574(2-(4-(6-Chloro-2-(4-methoxyphenyl)-3H-imidazo[4,5-...)
Affinity DataIC50:  52nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318568(2-(4-(6-Cyclopropyl-2-(4-methoxyphenyl)-3H-imidazo...)
Affinity DataIC50:  53nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318606((4-(6-Chloro-7-(4-((5-methylisoxazol-3-yl)methyl)p...)
Affinity DataIC50:  55nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318584(4-(6-Bromo-7-(4-(1-(pyridin-4-yl)ethyl)piperazin-1...)
Affinity DataIC50:  55nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318570(2-{4-[6-Bromo-2-(4-dimethylaminophenyl)-3H-imidazo...)
Affinity DataIC50:  55nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318579(2-(4-(6-Chloro-2-(4-(dimethylamino)phenyl)-3H-imid...)
Affinity DataIC50:  75nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318585(4-(6-chloro-7-(4-(1-phenylethyl)piperazin-1-yl)-3H...)
Affinity DataIC50:  79nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50335616(4-((4-(6-bromo-2-(4-methoxyphenyl)-3H-imidazo[4,5-...)
Affinity DataIC50:  81nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318571(2-[4-(6-Bromo-3H-imidazo[4,5-b]pyridin-7-yl)-piper...)
Affinity DataIC50:  81nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318573(2-[4-(6-Bromo-2-phenyl-3H-imidazo[4,5-b]pyridin-7-...)
Affinity DataIC50:  81nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318577(2-(4-(6-Chloro-2-(4-(dimethylamino)phenyl)-3H-imid...)
Affinity DataIC50:  115nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318578(2-(4-(6-Bromo-2-(4-(dimethylamino)phenyl)-3H-imida...)
Affinity DataIC50:  118nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318581(4-(6-Bromo-7-(4-(phenylsulfonyl)piperazin-1-yl)-3H...)
Affinity DataIC50:  178nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318583(4-(6-Bromo-7-(4-isobutylpiperazin-1-yl)-3H-imidazo...)
Affinity DataIC50:  210nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50224749(4-(6,7-dichloro-3H-imidazo[4,5-b]pyridin-2-yl)-N,N...)
Affinity DataIC50:  250nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318582(4-(6-Bromo-7-(4-phenylpiperazin-1-yl)-3H-imidazo[4...)
Affinity DataIC50:  258nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50335614(2-(4-(6-bromo-2-(4-(dimethylamino)phenyl)-3H-imida...)
Affinity DataIC50:  277nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50224745(4-(6-bromo-3H-imidazo[4,5-b]pyridin-2-yl)-N,N-dime...)
Affinity DataIC50:  490nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50224731(4-(6-chloro-3H-imidazo[4,5-b]pyridin-2-yl)-N,N-dim...)
Affinity DataIC50:  570nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50318593(6-Bromo-7-(4-cyclopropylmethyl-piperazin-1-yl)-2-(...)
Affinity DataIC50:  650nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50224742(2-(4-(2-(4-(dimethylamino)phenyl)-3H-imidazo[4,5-b...)
Affinity DataIC50:  870nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50224738(4-(7-chloro-3H-imidazo[4,5-b]pyridin-2-yl)-N,N-dim...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50224740(4-(3H-imidazo[4,5-b]pyridin-2-yl)-N,N-dimethylbenz...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50335613(2-(4-(pyridin-2-yl)phenyl)-3H-imidazo[4,5-b]pyridi...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50224736(2-(4-(pyrrolidin-1-yl)phenyl)-3H-imidazo[4,5-b]pyr...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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