TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
TargetEstrogen-related receptor gamma(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
TargetEstrogen-related receptor gamma(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
TargetEstrogen-related receptor gamma(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
TargetEstrogen-related receptor gamma(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
TargetEstrogen-related receptor gamma(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
TargetEstrogen-related receptor gamma(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.25E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
TargetEstrogen-related receptor gamma(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
TargetEstrogen-related receptor gamma(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
TargetEstrogen-related receptor gamma(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.78E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR2(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human ERRbeta ligand binding domain expressed in African green monkey CV1 cells assessed as...More data for this Ligand-Target Pair
TargetEstrogen-related receptor gamma(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
TargetEstrogen-related receptor gamma(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair
TargetEstrogen-related receptor gamma(Homo sapiens (Human))
The Beckman Research Institute
Curated by ChEMBL
The Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused mouse ERRgamma ligand binding domain expressed in African green monkey CV1 cells assessed a...More data for this Ligand-Target Pair