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Found 41 Enz. Inhib. hit(s) with all data for entry = 50035349
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123257(4-Benzhydryl-pyridine | CHEMBL150045)
Affinity DataKi:  79nMAssay Description:Affinity to displace binding of [3H]WIN-35428 to dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123256(4-(1,2-Diphenyl-ethyl)-pyridine | CHEMBL342055)
Affinity DataKi:  99nMAssay Description:Affinity to displace binding of [3H]WIN-35428 to dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM22418(Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...)
Affinity DataKi:  108nMAssay Description:Inhibition of [3H]DA uptake evaluated at the dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM22418(Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...)
Affinity DataKi:  155nMAssay Description:Inhibition of [3H]-5-HT uptake evaluated at the Serotonin transporterMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123257(4-Benzhydryl-pyridine | CHEMBL150045)
Affinity DataKi:  200nMAssay Description:Inhibition of reuptake of DA into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123257(4-Benzhydryl-pyridine | CHEMBL150045)
Affinity DataKi:  255nMAssay Description:Inhibition of [3H]DA uptake evaluated at the dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123256(4-(1,2-Diphenyl-ethyl)-pyridine | CHEMBL342055)
Affinity DataKi:  263nMAssay Description:Inhibition of [3H]DA uptake evaluated at the dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM22418(Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...)
Affinity DataKi:  270nMAssay Description:Affinity to inhibit [3H]DA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123256(4-(1,2-Diphenyl-ethyl)-pyridine | CHEMBL342055)
Affinity DataKi:  393nMAssay Description:Inhibition of [3H]-NE uptake evaluated at the monoamine transporter (NET)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123262(2-Benzhydryl-pyridine | CHEMBL347772)
Affinity DataKi:  742nMAssay Description:Affinity to displace binding of [3H]WIN-35428 to dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123255(3-Benzhydryl-pyridine | CHEMBL149246)
Affinity DataKi:  780nMAssay Description:Affinity to displace binding of [3H]WIN-35428 to dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123255(3-Benzhydryl-pyridine | CHEMBL149246)
Affinity DataKi:  860nMAssay Description:Inhibition of [3H]DA uptake evaluated at the dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123256(4-(1,2-Diphenyl-ethyl)-pyridine | CHEMBL342055)
Affinity DataKi:  910nMAssay Description:Inhibition of [3H]-5-HT uptake evaluated at the Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123266(3-(5-Naphthalen-2-yl-tetrazol-1-yl)-quinoline | CH...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of reuptake of DA into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123265(CHEMBL345273 | Diphenylvinylidene-methyl-amine)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of reuptake of DA into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123263(1-Benzyl-5-chloro-2-phenyl-1H-imidazole | CHEMBL14...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of reuptake of DA into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123269(3-Chloro-5,6-diphenyl-pyridazine-4-carbonitrile | ...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of reuptake of DA into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123267(3-(5-Phenyl-tetrazol-1-yl)-quinoline | CHEMBL14744...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of reuptake of DA into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123260(2-[(Z)-2-(2-Chloro-phenyl)-1-phenyl-vinyl]-pyridin...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of reuptake of DA into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123259(CHEMBL148615 | [Bis-(4-chloro-phenyl)-vinylidene]-...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of reuptake of DA into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123268(4-Dimethylamino-2,2-diphenyl-butyronitrile | CHEMB...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of reuptake of DA into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123262(2-Benzhydryl-pyridine | CHEMBL347772)
Affinity DataKi:  1.07E+3nMAssay Description:Inhibition of [3H]DA uptake evaluated at the dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123257(4-Benzhydryl-pyridine | CHEMBL150045)
Affinity DataKi:  1.16E+3nMAssay Description:Inhibition of [3H]-5-HT uptake evaluated at the Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123264(2,4-Dibenzyl-pyridine | CHEMBL147135)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of reuptake of DA into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123257(4-Benzhydryl-pyridine | CHEMBL150045)
Affinity DataKi:  3.46E+3nMAssay Description:Inhibition of [3H]-NE uptake evaluated at the monoamine transporter (NET)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123262(2-Benzhydryl-pyridine | CHEMBL347772)
Affinity DataKi:  5.53E+3nMAssay Description:Inhibition of [3H]-NE uptake evaluated at the monoamine transporter (NET)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123255(3-Benzhydryl-pyridine | CHEMBL149246)
Affinity DataKi:  7.32E+3nMAssay Description:Inhibition of [3H]-NE uptake evaluated at the monoamine transporter (NET)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123258(4-Anthracen-9-yl-pyridine | CHEMBL357312)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity to displace binding of [3H]WIN-35428 to dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123261(3-Anthracen-9-yl-pyridine | CHEMBL149878)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-5-HT uptake evaluated at the Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123261(3-Anthracen-9-yl-pyridine | CHEMBL149878)
Affinity DataKi: >1.00E+4nMAssay Description:Affinity to displace binding of [3H]WIN-35428 to dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123258(4-Anthracen-9-yl-pyridine | CHEMBL357312)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-5-HT uptake evaluated at the Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123254(4-Benzyl-pyridine | CHEMBL357322)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-NE uptake evaluated at the monoamine transporter (NET)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123254(4-Benzyl-pyridine | CHEMBL357322)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]DA uptake evaluated at the dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123254(4-Benzyl-pyridine | CHEMBL357322)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]DA uptake evaluated at the dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123254(4-Benzyl-pyridine | CHEMBL357322)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-5-HT uptake evaluated at the Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123261(3-Anthracen-9-yl-pyridine | CHEMBL149878)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-NE uptake evaluated at the monoamine transporter (NET)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123258(4-Anthracen-9-yl-pyridine | CHEMBL357312)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-NE uptake evaluated at the monoamine transporter (NET)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123261(3-Anthracen-9-yl-pyridine | CHEMBL149878)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]DA uptake evaluated at the dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123258(4-Anthracen-9-yl-pyridine | CHEMBL357312)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]DA uptake evaluated at the dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123255(3-Benzhydryl-pyridine | CHEMBL149246)
Affinity DataKi:  1.26E+4nMAssay Description:Inhibition of [3H]-5-HT uptake evaluated at the Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50123262(2-Benzhydryl-pyridine | CHEMBL347772)
Affinity DataKi:  3.50E+4nMAssay Description:Inhibition of [3H]-5-HT uptake evaluated at the Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed