Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with all data for entry = 50000146
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50241597(CHEMBL4074924)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged Brd4-BD1 expressed in Escherichia coli BL21(DE3) by LOGSY NMR titration methodMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50241596(CHEMBL4087267)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged Brd4-BD1 expressed in Escherichia coli BL21(DE3) by LOGSY NMR titration methodMore data for this Ligand-Target Pair